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Search Results for " Riluzole "

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カタログ番号 製品名 別名 ターゲット
T0349 Riluzole PK 26124,RP-54274 GABA Receptor , Sodium Channel , NMDAR
Riluzole (RP-54274) is a glutamate antagonist (RECEPTORS, GLUTAMATE) used as an anticonvulsant (ANTICONVULSANTS) and to prolong the survival of patients with AMYOTROPHIC LATERAL SCLEROSIS.
T37608 Riluzole-13C,15N2 Riluzole-13C,15N2
Riluzole-13C,15N2 is intended for use as an internal standard for the quantification of riluzole by GC- or LC-MS. Riluzole is a benzothiazole derivative with anti-excitotoxic effects that acts by blocking the presynaptic...
T41265 Riluzole hydrochloride
Riluzole hydrochloride, a use-dependent Na+ channel blocker with anticonvulsant properties, belongs to a category of drugs that also inhibit GABA uptake, exhibiting an inhibitory concentration 50 (IC50) of 43 μM.
T35919 N-hydroxy Riluzole
N-hydroxy Riluzole is a metabolite of the antiglutamatergic agent riluzole .1It is formed from riluzole predominantly by the cytochrome P450 (CYP) isoform CYP1A2 in human hepatic microsomes. 1.Sanderink, G.J., Bournique,...
T17174 Troriluzole BHV-4157 Others
Troriluzole is an orally active glutamate modulator. Troriluzole reduces the synaptic glutamate level and increases synaptic glutamate absorption.
T80626 VGSCs-IN-1 Sodium Channel
VGSCs-IN-1 is a potent VGSC inhibitor, a 2-piperazine analog of Riluzole that exhibits good blocking activity on Nav1.4.VGSCs-IN-1 can be used to study cellular excitability disorders.