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FDA-Approved Kinase Inhibitor Library

カタログ番号 L1610
  ライブラリー構成化合物リスト   Excel SDF

Kinases are a class of enzymes that facilitates phosphorylation, by transferring phosphate groups from high-energy donor molecules, such as ATP, to specific target molecules. A common group of kinases are the protein kinases, which act on specific proteins to phosphorylate them and alter their activity. Protein kinases are involved in a range of cell signaling and regulatory processes and play an important role in cell growth, metabolism, differentiation and apoptosis. Protein kinases have been associated with many diseases, including cancer, inflammatory diseases, cardiovascular diseases and neurological disorders. Therefore, targeting protein kinases has emerged as a promising therapeutic strategy for the treatment of related diseases.

Targetmol’s FDA-Approved Kinase Inhibitor Library contains 280 marketed drugs that target kinases. These kinases include Insulin/IGF Receptors、PI 3-Kinase、CaM Kinase II、JAK、PKA、CDK、JNK、PKC、CKI II、MAPK、RAF、EGFR、MEK、SAPK、GSK、MLCK、Src-family、IKK、PDGFR、VEGFR etc. FDA-Approved Kinase Inhibitor Library is a powerful tool for kinase drug development and related research.

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パッケージサイズ
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at [email protected]
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梱包・保管

  • バーコード付き貯蔵管や96/384-wellプレートに入っている粉末固体またはDMSO溶液
  • ブルーアイス同梱にて出荷
ライブラリ構成化合物複合リストをリクエスト (L1610)

Publications Cited TargetMol Libraries

隠し

ライブラリーの構成

Autophagy (72)
Apoptosis (57)
EGFR (35)
VEGFR (33)
c-Kit (32)
PDGFR (30)
FLT (18)
FGFR (18)
JAK (18)
Src (16)
Bcr-Abl (16)
Tyrosine Kinases (14)
c-Met/HGFR (14)
PKC (12)
CDK (12)
Raf (12)
ALK (11)
NF-κB (10)
Mitophagy (10)
Antibacterial (10)
AMPK (9)
PI3K (9)
c-RET (9)
Endogenous Metabolite (9)
BTK (8)
mTOR (8)
Adrenergic Receptor (8)
Antibiotic (8)
CaMK (8)
Sodium Channel (8)
5-HT Receptor (7)
MEK (7)
Ferroptosis (7)
PKA (7)
Trk receptor (7)
TAM Receptor (7)
ROCK (6)
ERK (6)
Potassium Channel (6)
Calcium Channel (6)
HER (6)
COX (5)
PDE (5)
HIV Protease (5)
ROS (5)
Histamine Receptor (5)
ROS Kinase (5)
Parasite (5)
Ras (5)
AChR (5)
Akt (5)
Dopamine Receptor (4)
p38 MAPK (4)
Serine/threonin kinase (4)
GSK-3 (4)
IκB/IKK (4)
Influenza Virus (4)
Antifungal (4)
P450 (3)
c-Fms (3)
IGF-1R (3)
Syk (3)
FAK (3)
SARS-CoV (3)
PAK (3)
Topoisomerase (3)
Glucosidase (3)
Phosphatase (2)
TNF (2)
Interleukin (2)
Serotonin Transporter (2)
DNA/RNA Synthesis (2)
MAPK (2)
P-gp (2)
Adenosine Receptor (2)
LPL Receptor (2)
Serine Protease (2)
Ephrin Receptor (2)
Nrf2 (2)
NADPH (2)
Glutathione Peroxidase (2)
TOPK (2)
Ligands for Target Protein for PROTAC (2)
Microtubule Associated (2)
PKM (2)
IRE1 (2)
Aurora Kinase (2)
ROR (2)
S1P Receptor (2)
Lipoxygenase (2)
Hexokinase (2)
Tyrosinase (2)
PLK (1)
JNK (1)
Proton pump (1)
Transferase (1)
Hydroxylase (1)
IFNAR (1)
DHFR (1)
HIF/HIF Prolyl-Hydroxylase (1)
HCV Protease (1)
Antioxidant (1)
Sigma receptor (1)
DNA-PK (1)
YAP (1)
Gap Junction Protein (1)
Dehydrogenase (1)
S6 Kinase (1)
Estrogen/progestogen Receptor (1)
Anti-infection (1)
Integrin (1)
NADPH-oxidase (1)
Mitochondrial Metabolism (1)
PPAR (1)
gp120/CD4 (1)
CSF-1R (1)
Monoamine Transporter (1)
Phosphorylase (1)
Reactive Oxygen Species (1)
GRK (1)
LDL (1)
Chloride channel (1)
HSV (1)
IL Receptor (1)
Chk (1)
PAD (1)
ACK (1)
GluR (1)
Norepinephrine (1)
DNA (1)
TRP/TRPV Channel (1)
HDAC (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Caspase (1)
TGF-beta/Smad (1)
Nucleoside Antimetabolite/Analog (1)
ATP Citrate Lyase (1)
AChE (1)
Antifolate (1)
Antiviral (1)
Hck (1)
Sirtuin (1)
HBV (1)
Melatonin Receptor (1)
Beta Amyloid (1)
Virus Protease (1)
NO Synthase (1)

化合物ライブラリー情報実例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE