ホーム 計算ツール
代理店ログイン

Anti-Metabolism Disease Compound Library

カタログ番号 L5200
  ライブラリー構成化合物リスト   Excel SDF

代謝は同化と異化からなる2つの反応に大別することができ、細胞および生物の生存状態を維持するための化学反応の集合であり、生体の恒常性を維持するための機能の1つです。代謝の研究における主眼は、生体制御機構とその肥満、糖尿病、心血管疾患、がんにおける役割です。

本製品は代謝疾患にフォーカスした1558の低分子化合物の独自のコレクションで、代謝に関連する研究および創薬スクリーニングに最適です。

TargetMolの製品は全て研究用試薬です。人体にはご使用できません。 また、個人の方への販売は行っておりません。
ご興味のある製品の価格と在庫は、こちらまでお問合せ下さい。
Get quote
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at [email protected]
ライブラリ構成化合物リストを依頼する
Get quote

製品概要

  • 1558種類の代謝関連化合物を独自にコレクション
  • ハイスループットスクリーニング(HTS)およびハイコンテンツスクリーニング(HCS)に最適
  • ほとんどが米国FDA、EMA、中国FDAの承認済み、臨床試験中、もしくは上市済み医薬品のため生物活性と安全性が確認済み
  • 糖尿病、肥満症、高トリグリセリド血症、高コレステロール血症などに関連する多様なターゲット(CYP、FAAH、IDO、MAOなど)をカバーする細胞代謝研究に有効なツール
  • 化合物の概要、化学構造、標的、IC50値、生物活性など詳細な情報を提供
  • 構造的多様性、薬効、細胞膜透過性を有する化合物
  • NMRとHPLCにより高純度と高品質を担保

ライブラリーのカスタマイズ

TargetMol社化合物ライブラリーは自由にカスタマイズできます! もっと詳しく

梱包・保管

  • バーコード付き貯蔵管や96/384-wellプレートに入っている粉末固体またはDMSO溶液
  • ブルーアイス同梱にて出荷
ライブラリ構成化合物複合リストをリクエスト (L5200)

ライブラリーの構成

Autophagy (241)
Apoptosis (189)
P450 (157)
Endogenous Metabolite (128)
Dehydrogenase (85)
AMPK (81)
Antibacterial (80)
PDE (77)
PPAR (72)
PI3K (55)
Antibiotic (51)
COX (49)
Glucocorticoid Receptor (39)
MAO (37)
Reactive Oxygen Species (37)
HSP (35)
HIV Protease (34)
Ferroptosis (32)
mTOR (32)
Parasite (31)
Potassium Channel (31)
FAAH (28)
Carbonic Anhydrase (27)
Akt (27)
NF-κB (27)
Lipoxygenase (26)
Calcium Channel (25)
Proteasome (25)
Antifungal (24)
Phosphatase (24)
Mitophagy (24)
GSK-3 (24)
Retinoid Receptor (23)
Phospholipase (23)
Influenza Virus (22)
RAAS (22)
DNA/RNA Synthesis (22)
Casein Kinase (21)
HIF/HIF Prolyl-Hydroxylase (20)
Mitochondrial Metabolism (20)
Monoamine Oxidase (20)
FXR (19)
DPP-4 (18)
NADPH (17)
Glucosidase (17)
ROCK (17)
5-HT Receptor (16)
CDK (16)
Transferase (16)
AChR (15)
Adrenergic Receptor (15)
HMG-CoA Reductase (15)
SARS-CoV (14)
GPR (14)
AhR (13)
HCV Protease (13)
Indoleamine 2,3-Dioxygenase (IDO) (13)
Reductase (13)
Sodium Channel (12)
PKA (12)
Adenosine Receptor (12)
IL Receptor (12)
Virus Protease (12)
Prostaglandin Receptor (12)
ATM/ATR (12)
ERK (11)
HIF (11)
MMP (11)
PARP (11)
Fatty Acid Synthase (11)
GABA Receptor (11)
HBV (11)
Glucokinase (11)
DHFR (11)
TNF (11)
Lipase (11)
SGLT (11)
Histamine Receptor (11)
S6 Kinase (11)
DNA-PK (11)
Wnt/beta-catenin (10)
transporter (10)
PKC (10)
Tyrosinase (10)
ROR (10)
Aryl Hydrocarbon Receptor (9)
ROS (9)
Cannabinoid Receptor (9)
Hydroxylase (9)
Caspase (9)
Serine Protease (9)
Liver X Receptor (9)
Estrogen/progestogen Receptor (9)
Estrogen Receptor/ERR (9)
PDK (8)
Glutathione Peroxidase (8)
Xanthine Oxidase (8)
NO Synthase (8)
ATPase (8)
Reverse Transcriptase (8)
HSV (8)
Dopamine Receptor (8)
Isocitrate Dehydrogenase (IDH) (8)
IκB/IKK (8)
Thrombin (8)
Interleukin (8)
JNK (8)
STAT (8)
NAMPT (8)
Factor Xa (8)
AChE (8)
Antifolate (8)
Nrf2 (7)
Stearoyl-CoA Desaturase (SCD) (7)
HDAC (7)
Cysteine Protease (7)
UGT (7)
PAI-1 (7)
Glucagon Receptor (7)
Lipid (7)
Topoisomerase (7)
IDO (7)
PKM (7)
Acyltransferase (6)
TRP/TRPV Channel (6)
Opioid Receptor (6)
P-gp (6)
Phosphorylase (6)
Neprilysin (6)
Sirtuin (6)
VEGFR (6)
Aminopeptidase (6)
Src (6)
BCL (5)
iGluR (5)
Beta Amyloid (5)
Microtubule Associated (5)
MEK (5)
SGK (5)
Androgen Receptor (5)
p38 MAPK (5)
c-Met/HGFR (5)
Chloride channel (5)
CETP (5)
FLT (5)
Serine/threonin kinase (4)
JAK (4)
CCR (4)
GluR (4)
NOS (4)
Aurora Kinase (4)
CAT (4)
Anti-infection (4)
Norepinephrine (4)
DNA (4)
CaMK (4)
Leukotriene Receptor (4)
ribosome (4)
LDL (4)
TGF-beta/Smad (4)
ATP Citrate Lyase (4)
GPCR19 (4)
RSV (4)
IGF-1R (3)
Carboxypeptidase (3)
Acetyl-CoA Carboxylase (3)
OAT (3)
Decarboxylase (3)
Thyroid hormone receptor(THR) (3)
Adiponectin receptor (3)
Hexokinase (3)
SIK (3)
Annexin A (3)
TAM Receptor (3)
P2Y Receptor (3)
Antioxidant (3)
ABC (3)
Integrin (3)
Drug Metabolite (3)
Antifection (3)
FGFR (3)
BACE (3)
c-RET (3)
PERK (3)
NADPH-oxidase (3)
Ras (3)
NPC1L1 (3)
MRP (3)
Vasopressin Receptor (3)
Endothelin Receptor (3)
Histone Demethylase (2)
Sigma receptor (2)
Trk receptor (2)
ASK (2)
Amino Acids and Derivatives (2)
LTR (2)
ALK (2)
Histone Methyltransferase (2)
ROS Kinase (2)
CFTR (2)
GST (2)
MLK (2)
p53 (2)
Proton pump (2)
Progesterone Receptor (2)
Chk (2)
Antiviral (2)
Nucleoside Antimetabolite/Analog (2)
Gap Junction Protein (2)
PDGFR (2)
EGFR (2)
E1/E2/E3 Enzyme (2)
Hedgehog/Smoothened (2)
Syk (2)
PAK (2)
Glutaminase (2)
cell cycle arrest (2)
Adenosine deaminase (2)
c-Kit (2)
Epigenetic Reader Domain (2)
MAPK (2)
Rho (2)
PGC-1α (2)
Tyrosine Kinases (2)
OX Receptor (2)
Epoxide Hydrolase (2)
Neurokinin receptor (2)
HER (1)
BMI-1 (1)
Complement System (1)
c-Fms (1)
CRISPR/Cas9 (1)
Aromatase (1)
cholecystokinin (1)
LPA Receptor (1)
PI4K (1)
DNA Methyltransferase (1)
Platelet aggregation (1)
DNA Alkylation (1)
MELK (1)
IFNAR (1)
IAP (1)
Serotonin Transporter (1)
Pim (1)
VDAC (1)
N-Acetylglucosaminyltransferase (1)
CaSR (1)
Galectin (1)
Melatonin Receptor (1)
Tie-2 (1)
RAR/RXR  (1)
DYRK (1)
aconitase (1)
DNA Alkylator/Crosslinker (1)
Immunology/Inflammation related (1)
LPL Receptor (1)
Arginase (1)
YAP (1)
DprE1 (1)
stilbene oxidase (1)
Hydrogenase (1)
Monocarboxylate transporter (1)
Transaminase (1)
GSNOR (1)
Adenylyl cyclase (1)
Mdm2 (1)
advanced glycation end products (1)
CSF-1R (1)
FLAP (1)
Pyroptosis (1)
Bradykinin Receptor (1)
hCE (1)
GluCls (1)
Free radical scavengers (1)
LRRK2 (1)
TLR (1)
Glutathione reductase (1)
PGE Synthase (1)
Beta-Secretase (1)
BCRP (1)
Telomerase (1)
PAD (1)
CXCR (1)
Thioredoxin (1)
RIP kinase (1)
Bombesin Receptor (1)
MAGL (1)
PROTAC Linker (1)
Smo (1)
Guanylate cyclase (1)
Anion Exchanger (1)
Monoamine Transporter (1)
DNA gyrase (1)
NMDAR (1)
MT Receptor (1)
GRK (1)
FABP (1)
Bcr-Abl (1)
S1P Receptor (1)

化合物ライブラリー情報実例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE