Powder: -20°C for 3 years | In solvent: -80°C for 1 year
AZD8329 is a selectable and potent inhibitor of human recombinant 11β-HSD1 and isolated human adipocyte 11ß-HSD1 and is an inhibitor of rat 11β-HSD1 (IC50 - 89nM) and dog recombinant 11β-HSD1. AZD8329 has a higher affinity for 11β-HSD1 than human recombinant 11β-HSD2 and 17 AZD8329 has the ability to reduce the activity of 11β-HSD1 in adipose tissue and liver samples.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約6-8 週間 | ¥ 176,000 |
50 mg | 約6-8 週間 | ¥ 228,500 |
100 mg | 約6-8 週間 | ¥ 399,500 |
説明 | AZD8329 is a selectable and potent inhibitor of human recombinant 11β-HSD1 and isolated human adipocyte 11ß-HSD1 and is an inhibitor of rat 11β-HSD1 (IC50 - 89nM) and dog recombinant 11β-HSD1. AZD8329 has a higher affinity for 11β-HSD1 than human recombinant 11β-HSD2 and 17 AZD8329 has the ability to reduce the activity of 11β-HSD1 in adipose tissue and liver samples. |
ターゲット&IC50 | 11β-HSD1 (human):9 nM |
分子量 | 421.53 |
分子式 | C25H31N3O3 |
CAS No. | 1048668-70-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 62.5 mg/mL (148.27 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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AZD8329 1048668-70-7 Metabolism Dehydrogenase AZD 8329 AZD-8329 Inhibitor inhibitor inhibit