Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
5 mg | 約6-8 週間 | ¥ 102,500 |
25 mg | 約6-8 週間 | ¥ 328,500 |
50 mg | 約6-8 週間 | ¥ 427,000 |
100 mg | 約6-8 週間 | ¥ 574,000 |
説明 | CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM). |
ターゲット&IC50 | Gastrin/CCK-A:1.82 μM , Gastrin/CCK-B:0.43 nM |
In vivo | CCK-B Receptor Antagonist 2 (0.1 μmol/kg; i.v.) has an inhibition effect on pentagastrin-induced gastric acid secretion in anesthetized rats (ED50: 8.3 nmol/kg). |
分子量 | 484.55 |
分子式 | C27H28N6O3 |
CAS No. | 155412-88-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL (515.94 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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CCK-B Receptor Antagonist 2 155412-88-7 Others CCK B Receptor Antagonist 2 CCKB Receptor Antagonist 2 Inhibitor inhibitor inhibit