Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CMPDA is a positive allosteric modulator of AMPA receptors (EC50s: 45.4 nM/63.4 nM for GluA2i/GluA2o receptor).
説明 | CMPDA is a positive allosteric modulator of AMPA receptors (EC50s: 45.4 nM/63.4 nM for GluA2i/GluA2o receptor). |
ターゲット&IC50 | GluA2i:45.4 nM (EC50), GluA2o:63.4 nM (EC50) |
In vitro | CMPDA was nearly equipotent at modulating the two isoforms of GluA2 receptors, whereas CMPDB displayed a modest preference for the flip splice variant. CMPDA slowed the rate of deactivation of GluA2o receptors approximately 2-fold but had no effect on GluA2i receptor deactivation. |
分子量 | 376.53 |
分子式 | C16H28N2O4S2 |
CAS No. | 380607-77-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Soluble
You can also refer to dose conversion for different animals. 詳細
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CMPDA 380607-77-2 Neuroscience GluR Inhibitor inhibitor inhibit