Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CP-96021 hydrochloride is a potent and orally active antagonist of leukotriene D4 (LTD4)/platelet activating factor receptor (Kis: 34 nM and 37 nM).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約8-10 週間 | ¥ 349,000 |
50 mg | 約8-10 週間 | ¥ 454,500 |
100 mg | 約8-10 週間 | ¥ 574,000 |
説明 | CP-96021 hydrochloride is a potent and orally active antagonist of leukotriene D4 (LTD4)/platelet activating factor receptor (Kis: 34 nM and 37 nM). |
ターゲット&IC50 | LTC4:34 nM (ki) |
In vivo | In vivo, CP-96021 inhibits iv LTD4- and iv PAF-induced bronchoconstriction in guinea pigs (ED50s: 0.46 and 0.16 mg/kg p.o.). CP-96021 effectively blocks the combined airway obstructive effects of endogenously released PAF and LTD4 stimulated by aerosolized antigen challenge in guinea pigs (ED50s: 1.8 mg/kg p.o.). |
分子量 | 529.03 |
分子式 | C29H22ClFN4OS |
CAS No. | 167011-22-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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CP-96021 hydrochloride 167011-22-5 Others CP-96021 Hydrochloride CP96021 hydrochloride CP 96021 hydrochloride CP96021 Hydrochloride CP 96021 Hydrochloride Inhibitor inhibitor inhibit