store at low temperature,store under nitrogen
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is an orally active and potent inhibitor of type I protein arginine methyltransferases (PRMTs) with anticancer and antitumor activity, inhibiting PRMT1, PRMT3, PRMT4, PRMT6, and PRMT8, and can be used to study advanced solid tumors.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
2 mg | 在庫あり | ¥ 18,500 | |||
5 mg | 在庫あり | ¥ 29,500 | |||
100 mg | 約10-14 週間 | ¥ 186,500 |
ターゲット&IC50 | PRMT3:48 nM, PRMT1:3.1 nM, PRMT6:5.7 nM, PRMT4:1148 nM, PRMT8:1.7 nM |
別名 | EPZ019997 dihydrochloride, GSK3368715 2HCl, EPZ019997 2HCl |
分子量 | 439.46 |
分子式 | C20H40Cl2N4O2 |
CAS No. | 1628925-77-8 |
store at low temperature,store under nitrogen
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: 100 mg/mL (227.55 mM), Sonication is recommended.
DMSO: 100 mg/mL (227.55 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
GSK3368715 dihydrochloride 1628925-77-8 Chromatin/Epigenetic Histone Methyltransferase EPZ019997 dihydrochloride GSK 3368715 GSK-3368715 Dihydrochloride EPZ-019997 EPZ 019997 Dihydrochloride GSK-3368715 GSK3368715 2HCl GSK3368715 Dihydrochloride EPZ 019997 EPZ019997 EPZ019997 2HCl EPZ-019997 Dihydrochloride GSK 3368715 Dihydrochloride GSK3368715 Inhibitor inhibitor inhibit