Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GW768505A free base is a potent dual inhibitor of VEGFR2 (KDR) and Tie-2 (pIC50: 7.81 for VEGFR2) with anti-angiogenic activity.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約6-8 週間 | ¥ 158,000 |
50 mg | 約6-8 週間 | ¥ 209,500 |
100 mg | 約6-8 週間 | ¥ 312,500 |
In vitro | GW768505A free base acts as an inhibitor of both KDR and TIE2, demonstrating significant inhibition (71–88% inhibition at 100 nM) of tropomyosin-related kinases, including TRKA, TRKB, and TRKC. Furthermore, it exhibits inhibitory effects on the growth of cancer cells in the NCI-60 panel screening. |
分子量 | 537.47 |
分子式 | C27H19F4N5O3 |
CAS No. | 501693-25-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
GW768505A free base 501693-25-0 Others GW768505A GW-768505A free base Inhibitor inhibitor inhibit