keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Kinetensin acetate(103131-69-7 free base) is isolated from pepsin-treated human plasma. Kinetensin acetate(103131-69-7 free base) is a neurotensin-like peptide.
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1 mg | 在庫あり | ¥ 22,000 | |||
5 mg | 在庫あり | ¥ 43,500 | |||
10 mg | 在庫あり | ¥ 70,500 | |||
25 mg | 在庫あり | ¥ 124,000 | |||
50 mg | 在庫あり | ¥ 179,000 | |||
100 mg | 在庫あり | ¥ 250,500 |
説明 | Kinetensin acetate(103131-69-7 free base) is isolated from pepsin-treated human plasma. Kinetensin acetate(103131-69-7 free base) is a neurotensin-like peptide. |
In vitro | The peptide kinetensin isolated from pepsin-treated human plasma induces a dose-dependent release of histamine when exposed to rat peritoneal mast cells. The threshold concentration is around 1 μM, the ED50 is 10 μM, and the optimal concentration of between 100 to 1000 μM released 80% of the total histamine. Kinetensin is 10 to 100 times less potent than neurotensin and equipotent with the opioid peptide dynorphin. The histamine release is clearly temperature-dependent, with no release occurring at 0 or 45 °C and with an optimum around 37 °C. The histamine release is significantly reduced in the absence of extracellular calcium[2]. |
In vivo | Kinetensin also induces a dose-dependent increase in vascular permeability when injected intradermally into rats[2]. |
別名 | Kinetensin (human) acetate |
分子量 | 1232.45 |
分子式 | C58H89N17O13 |
CAS No. | TP1116L |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 10 mM
You can also refer to dose conversion for different animals. 詳細
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Kinetensin acetate(103131-69-7 free base) TP1116L GPCR/G Protein Neurotensin Receptor Kinetensin acetate(103131697 free base) Kinetensin Kinetensin Acetate Kinetensin (human) acetate Kinetensin acetate(103131 69 7 free base) Inhibitor inhibitor inhibit