Powder: -20°C for 3 years | In solvent: -80°C for 1 year
L-692429 (MK-0751) is a potent nonpeptidyl growth hormone secretagogue (GHS) agonist, a benzolactam derivative, which reverses the inhibition of GH secretion by glucocorticoids.L-692429 has a high affinity for the G protein-coupled receptor and can be used in the study of acromegaly and obesity. L-692429 has a high affinity for G protein-coupled receptor and can be used to study acromegaly and obesity.
ターゲット&IC50 | intracellular calcium:26 nM (EC50), BRET:58 nM (EC50), inositol phosphate (IP) turnover:47 nM (EC50), Serum-responsive element activity:63 nM (EC50), CREB:60 nM (EC50) |
別名 | MK-0751 |
分子量 | 509.614 |
分子式 | C29H31N7O2 |
CAS No. | 145455-23-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 40 mg/mL (78.49 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
L-692429 145455-23-8 GPCR/G Protein GHSR GPCR19 MK 0751 L692429 MK0751 MK-0751 L 692429 Inhibitor inhibitor inhibit