Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Lp-PLA2-IN-2 is a selective and potent lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor, with an IC50 0f 120 nM for recombinant human Lp-PLA2.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約8-10 週間 | ¥ 486,500 |
50 mg | 約8-10 週間 | ¥ 638,000 |
100 mg | 約8-10 週間 | ¥ 849,500 |
説明 | Lp-PLA2-IN-2 is a selective and potent lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor, with an IC50 0f 120 nM for recombinant human Lp-PLA2. |
ターゲット&IC50 | Lp-PLA2:120 nM |
In vitro | Lp-PLA2-IN-2 inhibits Human Lp-PLA2 with an IC50 of 62 nM in PED6 assay. |
In vivo | Lp-PLA2-IN-2 (1 mg/kg;?i.v.) treament in rats shows that the Cl, Vss and t1/2 values are 67 mL/min/kg, 1.2 L/kg, and 0.34 hours, respectively[1]. |
分子量 | 394.46 |
分子式 | C19H23FN2O4S |
CAS No. | 2071636-15-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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Lp-PLA2-IN-2 2071636-15-0 Metabolism Phospholipase LpPLA2IN2 Lp-PLA-2-IN-2 Lp PLA2 IN 2 Inhibitor inhibitor inhibit