Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. Mavoglurant (racemate) is the racemate of mavoglurant.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約6-8 週間 | ¥ 349,000 |
50 mg | 約6-8 週間 | ¥ 454,500 |
100 mg | 約6-8 週間 | ¥ 574,000 |
説明 | Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. Mavoglurant (racemate) is the racemate of mavoglurant. |
In vitro | For antagonistic activity, (?)-mavoglurant, the (?)-enantiomer shows IC50 of 0.11 μM and 0.03 μM (Ca2+ and PI-turnover) whereas the (+)-enantiomer ((+)-10) shows only 37% and 18% inhibition at 10 μM. |
別名 | AFQ-056 racemate |
分子量 | 313.39 |
分子式 | C19H23NO3 |
CAS No. | 1636881-61-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (159.55 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Mavoglurant racemate 1636881-61-2 Others AFQ-056 racemate Inhibitor inhibitor inhibit