Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Mps1-IN-1 is a potent, selective and ATP-competitive inhibitor of Mps1 kinase (IC50 : 367 nM )
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 9,000 | |||
5 mg | 在庫あり | ¥ 21,000 | |||
10 mg | 在庫あり | ¥ 39,000 | |||
25 mg | 在庫あり | ¥ 76,500 | |||
50 mg | 在庫あり | ¥ 114,500 | |||
100 mg | 在庫あり | ¥ 166,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 24,500 |
説明 | Mps1-IN-1 is a potent, selective and ATP-competitive inhibitor of Mps1 kinase (IC50 : 367 nM ) |
ターゲット&IC50 | FAK:440 nM (kd), CLK1:1900 nM (kd), TYK1/LTK:29 nM (kd), PYK2:280 nM (kd), TNK1:2600 nM (kd), ERK2:2900 nM (kd), ALK:21 nM (kd), INSR:470 nM (kd), IGF-1R:750 nM (kd), Mps1:27 nM (kd), GAK:1100 nM (kd), TNK2:3100 nM (kd), INSRR:1200 nM (kd) |
In vitro | Mps1-IN-1 is a potent, selective and ATP-competitive inhibitor of Mps1 kinase(IC50 and a Kd of 367 nM and 27 nM). Mps1-IN-1 also has high affinity for ALK, and LTK, with Kds of 21 and 39 nM, respectively[1]. |
分子量 | 535.66 |
分子式 | C28H33N5O4S |
CAS No. | 1125593-20-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 39 mg/mL (72.81 mM)
You can also refer to dose conversion for different animals. 詳細
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Mps1-IN-1 1125593-20-5 Others Mps-1-IN-1 Mps1IN1 Mps1 IN 1 Inhibitor inhibitor inhibit