Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PCSK9 ligand 1 is a small molecule ligand for proprotein convertase substilisin-like/kexin type 9 (PCSK9) and shows high affinity to PCSK9(Ki of 107 nM).
説明 | PCSK9 ligand 1 is a small molecule ligand for proprotein convertase substilisin-like/kexin type 9 (PCSK9) and shows high affinity to PCSK9(Ki of 107 nM). |
ターゲット&IC50 | PCSK9(ki):ki:107 nM |
In vitro | PCSK9 ligand 1 treatment shows a clear concentration-dependent degradation of both the pro and mature form of PCSK9 yielding a half-maximal degradation concentration of 4.8 and 3.4 μM, as well as a maximum percentage of degradation at 20 μM of 58% and 61%, respectively[1]. |
分子量 | 1077.22 |
分子式 | C53H69FN8O13S |
CAS No. | 2216703-12-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
PCSK9 ligand 1 2216703-12-5 Others PCSK-9 ligand 1 Inhibitor inhibitor inhibit