Powder: -20°C for 3 years | In solvent: -80°C for 1 year
SGK1-IN-1 is a highly active and selective SGK-1 inhibitor(IC50 of 1 nM).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
2 mg | 約 5 days | ¥ 53,500 |
5 mg | 約 5 days | ¥ 68,500 |
25 mg | 約6-8 週間 | ¥ 226,500 |
50 mg | 約6-8 週間 | ¥ 312,500 |
100 mg | 約6-8 週間 | ¥ 427,000 |
ターゲット&IC50 | SGK1:1 nM |
In vitro | SGK1-IN-1 (14n) demonstrates favorable SGK isoform selectivity, exhibiting potent activity towards hSGK2 and moderate activity against hSGK3, with IC50 values of 1 and 41 nM at ATP concentrations of 10 μM and 50 μM, respectively. Additionally, it shows cellular efficacy by inducing SGK1-dependent phosphorylation of GSK3β in U2OS cells, achieving an activity level of 0.69 μM[2]. |
分子量 | 418.83 |
分子式 | C17H12ClFN6O2S |
CAS No. | 1279829-87-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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SGK1-IN-1 1279829-87-6 Others SGK1IN1 SGK1 IN 1 SGK-1-IN-1 Inhibitor inhibitor inhibit