keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Taspoglutide is a long-acting glucagon-like peptide 1 (GLP-1) receptor agonist(EC50 value of 0.06 nM),and for treatment of type 2 diabetes
ターゲット&IC50 | GLP1:(EC50)0.06 nM |
In vitro | Taspoglutide (R1583/BIM51077), exhibiting 93% homology with native polypeptides, is a long-acting formulation of (Aib8-35) human GLP-1 (7-36 amides) that activates the GLP-1 receptor. It demonstrates an affinity constant (1.1±0.2 nM) towards the hGLP-1 receptor, closely mirroring the natural ligand’s affinity constant of 1.5±0.3 nM, and shows similar potency in stimulating cAMP production [2]. |
別名 | R1583, BIM51077, ITM077 |
分子量 | 3339.763 |
分子式 | C152H232N40O45 |
CAS No. | 275371-94-3 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 28 mg/mL (8.38 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Taspoglutide 275371-94-3 Others R 1583 R-1583 R1583 BIM 51077 ITM 077 BIM-51077 BIM51077 ITM-077 ITM077 Inhibitor inhibitor inhibit