Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ciprostene is the 9β-methyl analog of carbaprostacyclin and a stable analog of PGI2. Ciprostene exhibits biological activity similar to PGI2, but is 30-fold less potent. In patas monkeys, ciprostene induces hypotension and causes tachycardia when administered at a dose of 0.16 μg/kg/min. In addition, ciprostene inhibits ADP-induced platelet aggregation ex vivo and in vitro with ID50 values of 9.1 μg/kg/min and 60 ng/ml, respectively.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 約 35 days | ¥ 87,500 |
5 mg | 約 35 days | ¥ 388,000 |
10 mg | 約 35 days | ¥ 675,000 |
説明 | Ciprostene is the 9β-methyl analog of carbaprostacyclin and a stable analog of PGI2. Ciprostene exhibits biological activity similar to PGI2, but is 30-fold less potent. In patas monkeys, ciprostene induces hypotension and causes tachycardia when administered at a dose of 0.16 μg/kg/min. In addition, ciprostene inhibits ADP-induced platelet aggregation ex vivo and in vitro with ID50 values of 9.1 μg/kg/min and 60 ng/ml, respectively. |
分子量 | 771.146 |
分子式 | C44H74CaO8 |
CAS No. | 81703-55-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PBS (pH 7.2): > 0.29 μg/mL
DMSO: > 16.8 mg/mL
DMF: > 25 mg/mL
Ethanol: > 34 mg/mL
You can also refer to dose conversion for different animals. 詳細
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Ciprostene (calcium salt) 81703-55-1 Ciprostene Inhibitor inhibitor inhibit