Powder: -20°C for 3 years | In solvent: -80°C for 1 year
HDAC6/8/BRPF1-IN-1 is a dual inhibitor that targets HDAC6, HDAC8, and the bromodomain and PHD finger containing protein 1 (BRPF1). It exhibits inhibitory activity against HDAC1, HDAC6, and HDAC8 with IC50 values of 797 nM, 344 nM, and 908 nM, respectively. In addition, it inhibits BRPF1 with a Kd value of 175.2 nM. This compound is utilized in cancer research [1].
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約6-8 週間 | ¥ 349,000 |
50 mg | 約6-8 週間 | ¥ 454,500 |
100 mg | 約6-8 週間 | ¥ 574,000 |
説明 | HDAC6/8/BRPF1-IN-1 is a dual inhibitor that targets HDAC6, HDAC8, and the bromodomain and PHD finger containing protein 1 (BRPF1). It exhibits inhibitory activity against HDAC1, HDAC6, and HDAC8 with IC50 values of 797 nM, 344 nM, and 908 nM, respectively. In addition, it inhibits BRPF1 with a Kd value of 175.2 nM. This compound is utilized in cancer research [1]. |
In vitro | HDAC6/8/BRPF1-IN-1 exhibits inhibitory activity against HDAC1, HDAC6, and HDAC8, with IC50 values of 797 nM, 344 nM, and 908 nM, respectively, and demonstrates inhibition of BRPF1 with a Kd value of 175.2 nM [1]. |
分子量 | 387.41 |
分子式 | C18H17N3O5S |
CAS No. | 2484255-65-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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HDAC6/8/BRPF1-IN-1 2484255-65-2 Inhibitor inhibitor inhibit