keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
K41498 acetate, an analogues of antisauvagine-30 (aSvg-30), inhibits sauvagine-stimulated cAMP accumulation in hCRF2α- and hCRF2β-expressing cells. K41498 acetate is a potent and highly selective antagonist CRF2 receptor with Ki values of 0.66 nM, 0.62 nM and 425 nM for human CRF2α, CRF2β and CRF1 receptors respectively.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 143,000 |
5 mg | 在庫あり | ¥ 305,500 |
10 mg | 在庫あり | ¥ 408,500 |
25 mg | 在庫あり | ¥ 615,000 |
50 mg | 在庫あり | ¥ 824,000 |
100 mg | 在庫あり | ¥ 1,120,000 |
説明 | K41498 acetate, an analogues of antisauvagine-30 (aSvg-30), inhibits sauvagine-stimulated cAMP accumulation in hCRF2α- and hCRF2β-expressing cells. K41498 acetate is a potent and highly selective antagonist CRF2 receptor with Ki values of 0.66 nM, 0.62 nM and 425 nM for human CRF2α, CRF2β and CRF1 receptors respectively. |
ターゲット&IC50 | CRF2α:0.66 nM(Ki), CRF2β:0.62 nM(Ki), CRF1:425 nM(Ki) |
分子量 | N/A |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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K 41498 aceate GPCR/G Protein CRFR Inhibitor inhibitor inhibit