Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PSN 375963 hydrochloride, a potent GPR119 agonist, demonstrates EC50 values of 8.4 μM and 7.9 μM for human and mouse GPR119, respectively. Its efficacy is comparable to that of the endogenous agonist oleoylethanolamide (OEA) [1] [2].
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約6-8 週間 | ¥ 349,000 |
50 mg | 約6-8 週間 | ¥ 454,500 |
100 mg | 約6-8 週間 | ¥ 574,000 |
説明 | PSN 375963 hydrochloride, a potent GPR119 agonist, demonstrates EC50 values of 8.4 μM and 7.9 μM for human and mouse GPR119, respectively. Its efficacy is comparable to that of the endogenous agonist oleoylethanolamide (OEA) [1] [2]. |
In vitro | The endogenous ligand oleoylethanolamide (OEA) activates GPR119 in a way comparable to the interaction of glucagon-like peptide-1 (GLP-1) with its receptor, influencing insulin secretion, intracellular calcium levels, and cyclic AMP concentration [2]. |
分子量 | 321.85 |
分子式 | C17H24ClN3O |
CAS No. | 1781834-82-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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PSN 375963 hydrochloride(388575-52-8 Free base) 1781834-82-9 Others PSN-375963 Hydrochloride 388575-52-8 PSN 375963 Hydrochloride PSN 375963 hydrochloride(388575 52 8 Free base) PSN 375963 hydrochloride(388575528 Free base) 388575-52-8 Free base PSN375963 Hydrochloride Inhibitor inhibitor inhibit