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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T61197 | Irdabisant hydrochloride | Others | |
Irdabisant hydrochloride (CEP-26401) is a selective, orally active, and blood-brain barrier (BBB) penetrant histamine H3 receptor (H3R) inverse agonist/inverse agonist, demonstrating high affinity with K*i values of 7.2 ... | |||
T32191 | Irdabisant | CEP-26401,CEP 26401,CEP26401 | Histamine Receptor |
Irdabisant (CEP-26401) (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R) (rat H3R Ki= 7.2 nM, human H3R Ki= 2.0 nM). Irdabisant ex... |