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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T62621 | Pan-HER-IN-2 | Others | |
pan-HER-IN-2 (Compound C6) is an orally active, reversible, broad-spectrum HER inhibitor that acts on EGFR (IC50: 0.72 nM), HER4 (IC50: 2.0 nM), EGFRT790M (IC50: 8.2 nM), and L858R (IC50: 75.1 nM). pan-HER-IN-2 induces a... |