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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T12861 | SB-277011 | SB-277011A | Dopamine Receptor |
SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and 5-HT1B respectively. | |||
T12861L | SB-277011 dihydrochloride | SB-277011A dihydrochloride | Dopamine Receptor |
SB-277011 dihydrochloride is a potent, selective, orally bioavailable and brain penetrate antagonist of dopamine D3 receptor(pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively). | |||
T63096 | SB-277011 hydrochloride | ||
SB-277011 hydrochloride (SB-277011A hydrochloride) is a potent, selective, orally active, dopamine D3 receptor (D3R) antagonist that crosses the blood-brain barrier with Ki values of 10.7 nM and 11.2 nM for rodent and hu... |