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T1049L |
Oxybutynin
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Oxytrol,Ditropan,Oxibutyninum |
Potassium Channel
,
AChR
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Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome. |
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T1049 |
Oxybutynin chloride
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Oxybutynin hydrochloride,Oxybutynin HCl |
Potassium Channel
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AChR
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Oxybutynin chloride (Oxybutynin HCl) is an anticholinergic medication used to relieve urinary and bladder difficulties. It competitively antagonizes the M1, M2, and M3 subtypes of the muscarinic acetylcholine receptor. |
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T70139 |
MSD-D
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Others
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MSD-D is an inhibitor of voltage-gated K(+) (Kv) channels Kv1.5. |
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T80054 |
Phrixotoxin 2
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Potassium Channel
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Phrixotoxin 2 selectively blocks the KV 4.2 and KV 4.3 channels, demonstrating high specificity in its interaction with these voltage-gated ion channels [1]. |
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T37808 |
Kaliotoxin
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Kaliotoxin is an inhibitor of neuronal BK-type peptide groups and specifically inhibits Kv channels and calcium-activated potassium channels. Kaliotoxin has research significance on the regulation of cell membrane potent... |
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T36803 |
AAQ chloride
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Others
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Photoswitchable Kv channel blocker (IC50 values are 2 and 64 μM at 500 nm and 380 nm respectively). Switches conformation from cis to trans at 500 nm and trans to cis at 380 nm. Exhibits minimal activity at Nav1.2 and L-... |
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T84382 |
LY303511 hydrochloride
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Others
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LY303511, a structural analog of LY294002, selectively inhibits mTOR-dependent phosphorylation of S6K, unlike its counterpart, which acts as a phosphatidylinositol 3-kinase (PI3K) inhibitor. It effectively reduces cell p... |
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T36066 |
NADP+ (sodium salt hydrate)
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Others
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NADP+ is the oxidized form of the electron donor nicotinamide adenine dinucleotide phosphate . It serves as a cofactor in various biological reactions. In addition, the balance between these reduced and oxidized forms pl... |
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T84443 |
Halofuginone hydrochloride
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RU-19110 hydrochloride |
Others
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Halofuginone hydrobromide (RU-19110), a derivative of Febrifugine, functions as a competitive inhibitor of prolyl-tRNA synthetase, displaying a K_i value of 18.3 nM. This compound effectively inhibits type-I collagen syn... |
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T80483 |
Aam-KTX
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Potassium Channel
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Aam-KTX, a toxic peptide sourced from Mesobuthus eupeus scorpion venom, acts as a selective K_v channel inhibitor, exhibiting IC_50 values of 1.1 nM for K_v1.3 channels and >750 nM for K_v1.1 channels. This compound show... |
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T80851 |
VSTx-3
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Kappa-TRTX-Gr4a,κ-Theraphotoxin-Gr4a,Voltage sensor toxin 3,Peptide F |
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VSTx-3 is a potassium voltage-gated channel (K_V) blocker, which has also been shown to be a potent tetrodotoxin-sensitive (TTX-sensitive) sodium channel inhibitor, with particular efficacy against NaV1.8 channels, as ev... |
