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カタログ番号 | 製品名 | 別名 | ターゲット |
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T24941 | VMAT2-IN-I HCl | VMAT2 IN I Hydrochloride,VMAT2-IN-I Hydrochloride,VMAT2INI Hydrochloride | |
VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A. | |||
T79061 | VMAT2-IN-2 tosylate | Monoamine Transporter | |
VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1]. | |||
T7147 | Valbenazine | NBI-98854 | Monoamine Transporter |
Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia. | |||
T0719 | Tetrabenazine | Xenazine,Ro 1-9569 | Others , Dopamine Receptor , Monoamine Transporter |
Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders. Tetrabenazine blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high... | |||
T7563 | NBI-98782 | (+)-α-Dihydrotetrabenazine,(+)-α-DHTBZ,(+)-DTBZ | Monoamine Transporter |
NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM) | |||
T13133 | Tetrabenazine Metabolite | (-)-β-Dihydrotetrabenazine,(-)-β-HTBZ | Monoamine Transporter |
Tetrabenazine Metabolite ((-)-β-HTBZ), a vesicles monoamine transporter 2 (VMAT2) inhibitor, is an active metabolite of Tetrabenazine. Tetrabenazine Metabolite has a high affinity for VMAT2 with a Ki of 13.4 nM. Tetraben... | |||
T41195 | FFN 206 dihydrochloride | ||
FFN 206 dihydrochloride is a fluorescent VMAT2 substrate that can be used to detect VMAT2 subcellular sites in cell culture and shows no detectable inhibition of DAT. | |||
T13134 | (+)-Tetrabenazine | (+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ | Monoamine Transporter |
(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1. | |||
T41194 | FFN 102 mesylate | Others | |
FFN 102 mesylate is a pH responsive fluorescent false neurotransmitter (FFN), a selective dopamine transporter (DAT) and VMAT2 substrate. Exhibits no significant binding to a panel of 38 CNS receptors, including dopamine... | |||
T77549 | Nurr1 agonist 2 | Others | |
Nurr1 agonist 2 is a Nurr1 agonist with an EC50 value of 0.07 μM. Nurr1 agonist 2 increases the mRNA expression of the Nurr1-regulated genes tyrosine hydroxylase (TH) and vesicular amino acid transporter 2 (VMAT2). Nurr1... | |||
T22452 | Valbenazine tosylate | NBI-98854 | Monoamine Transporter |
Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM). | |||
T25750 | Lobelane Hydrochloride | ||
Lobelane Hydrochloride is a vesicular monoamine transporter-2 (VMAT2) inhibitor. | |||
T31791 | FFN246 HCl | FFN 246,FFN246 hydrochloride,FFN246,FFN-246 | |
FFN246 is a fluorescent substrate for both the serotonin transporter and the vesicular monoamine transporter 2 (VMAT2). | |||
T70322 | Valbenazine dihydrochloride | ||
Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia. | |||
T12190 | Trans (2,3)-Dihydrotetrabenazine | (2R,3R,11bR)-rel-DHTBZ,(2R,3R,11bR)-rel-Dihydrotetrabenazine | Others |
Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2). | |||
T31790 | FFN200 dihydrochloride | FFN200 HCl,FFN200,FFN 200,FFN-200 | |
FFN200 is a vesicular monoamine transporter 2 (VMAT2) substrate that selectively traces monoamine exocytosis in both neuronal cell culture and brain tissue. | |||
T23983 | Deutetrabenazine metabolite M4 | SD-1018,Deuterated monohydroxy tetrabenazine,D6-tetrabenazine metabolite M4 | |
Deutetrabenazine metabolite M4 is believed to be related to its effect as a reversible depletion of monoamines from nerve terminals. The major circulating metabolites of Deutetrabenazine, are reversible inhibitors of VM... | |||
T78684 | FFN246 | 5-HT Receptor | |
FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation and emission spectra at 392/427 nm, respectively. It serves to label... | |||
T41193 | FFN 270 | ||
FFN 270 is a fluorescent false neurotransmitter (FFN). Fluorescent substrate for NET and VMAT2. Labels noradrenergic neurons and their synaptic vesicles, and enables imaging of synaptic vesicle content release from speci... |