2
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T2588 | Ivacaftor | Ivacaftor (VX-770),VX-770 | CFTR , Autophagy |
Ivacaftor (VX-770) (VX-770) is a potentiator of CFTR targeting G551D-CFTR (EC50: 100 nM) and F508del-CFTR (EC50: 25 nM) in Fisher rat thyroid cells, respectively. | |||
T13742L | Ivacaftor hydrate | VX-770 hydrate | Others |
Ivacaftor hydrate is an orally bioavailable CFTR potentiator. It also is used for cystic fibrosis treatment. |