5
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T2326 | Tolvaptan | OPC-41061 | Vasopressin Receptor , Autophagy |
Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia. | |||
T6288 | Mozavaptan | OPC31260l,OPC-31260 | Vasopressin Receptor |
Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively. | |||
T6453 | Conivaptan hydrochloride | Vaprisol,Conivaptan HCl,YM 087 | Vasopressin Receptor |
Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic. | |||
T73660 | ZP 120C | ||
ZP 120C, a potent and partial ORL1 receptor agonist, effectively inhibits electrically induced contraction. It is utilized in the research of hyponatremia/hypokalemia [1] [3]. | |||
T21378 | Conivaptan | YM087,YM-087,YM 087,Vaprisol | |
Conivaptan, a non-peptide inhibitor of antidiuretic hormone, was approved for hyponatremia caused by the syndrome of inappropriate antidiuretic hormone (SIADH), there is also some evidence that it may be effective in hea... |