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c-Myc

Myc is a family of regulator genes and proto-oncogenes that code for transcription factors. The Myc family consists of three related human genes: c-myc (MYC), l-myc (MYCL), and n-myc (MYCN). c-myc (also sometimes referred to as MYC) was the first gene to be discovered in this family, due to homology with the viral gene v-myc.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T3686 10074-G5 413611-93-5 98%
10074-G5 is an inhibitor of c-Myc-Max dimerization.
T12133 MYCi975 2289691-01-4 98%
MYCi975 (NUCC-0200975) is an orally active inhibitor of MYC.
T12132 MYCi361 2289690-31-7 98%
MYCi361 (NUCC-0196361) is an inhibitor of MYC (binding to MYC with Kd of 3.2 μM).
TN6508 Trachelogenin 34209-69-3 98%
Trachelogenin ((-)-Trachelogenin), an HCV entry inhibitor, has antiproliferative effects, and its mechanism is related to affecting the phosphorylation of key pr...
T9628 10074-A4 312631-87-1 98%
10074-A4 is a c-Myc binding compound that associates with c-Myc370–409 and behaves like a “ligand cloud” around a “protein cloud”, with distinct features from th...
T15665 KJ Pyr 9 581073-80-5
KJ Pyr 9 is an MYC inhibitor (Kd: 6.5 nM in vitro assay).
T12134 MYCMI-6 681282-09-7 97.77%
MYCMI-6 (NSC-354961) is a potent and selective inhibitor of endogenous MYC:MAX protein interactions,reduces proliferation and induces massive apoptosis in tumor ...
T9033 BTYNB 304456-62-0 98%
BTYNB (MDK6620) is an inhibitor of the oncofetal mRNA-binding protein IMP1 (IC50 = 5 μM for IMP1 binding to c-Myc mRNA). MDK6620 downregulates β-TrCP1 mRNA and r...
T9061 EN4 1197824-15-9 98.19%
EN4 (EN4 MYC inhibitor) MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It is selective for c-MYC over N-MYC and L-MYC, and inhibits ...
TN1892 Lusianthridin 87530-30-1 99.11%
Lusianthridin is a natural product from Dendrobium venustum. Lusianthridin exhibits anti-migratory property at nontoxic concentrations. Lusianthridin enhances c-...
T10352 APTO-253 916151-99-0 99.43%
APTO-253 (LOR-253) inhibits c-Myc expression, stabilizes G-quadruplex DNA, and induces cell cycle arrest and apoptosis in acute myeloid leukemia cells. APTO-253 ...
T4252 ML327 1883510-31-3 99.48%
ML327 is a MYC blocker. ML327 can also de-repress E-cadherin transcription and reverse Epithelial-to-Mesenchymal Transition (EMT).
T4367 Mycro 3 944547-46-0 99.51%
Mycro 3 is potent and selective for c-Myc in whole cell assays.
T9093 NY2267 886053-73-2 99.6%
NY2267 (Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl ester...
T3048 10058-F4 403811-55-2 99.82%
10058-F4 (c-Myc Inhibitor) is a cell-permeable thiazolidinone that specifically inhibits the c-Myc-Max interaction and prevents transactivation of c-Myc target g...
T0617 Nicotinamide N-oxide 1986-81-8 99.9%
Nicotinamide N-oxide (Nicotinamide 1-oxide) is recognized as an in vivo metabolite of nicotinamide which is a precurser of nicotinamide-adenine dinucleotide (NAD...
T60019 VPC-70063 13571-44-3 99.93%
VPC-70063 (Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)-) is an inhibitor of c-Myc-MAX. VPC-70063 exhibits Myc-Max transcriptional activity inh...
TN4581 Moracin D 69120-07-6 98%
Moracin C and moracin D, new phytoalexins from diseased mulberry, are antifungal compounds. Moracin may be protective influence in tumor promotion, utilization o...
T10702 CBP/p300-IN-2 2158265-96-2 98%
CBP/EP300-IN-2 is an inhibitor of CBP/EP300 (IC50s: 1.07 nM and 5.96 nM for CBP/HTRF and Myc) extracted from patent WO2017205538A1 (example 25).
TN1354 Aaptamine 85547-22-4 98%
Aaptamine functions as a proteasome inhibitor, it activates p21 promoter in a p53-independent manner.
10074-G5
T3686
10074-G5 is an inhibitor of c-Myc-Max dimerization.
MYCi975
T12133
MYCi975 (NUCC-0200975) is an orally active inhibitor of MYC.
MYCi361
T12132
MYCi361 (NUCC-0196361) is an inhibitor of MYC (binding to MYC with Kd of 3.2 μM).
Trachelogenin
TN6508
Trachelogenin ((-)-Trachelogenin), an HCV entry inhibitor, has antiproliferative effects, and its mechanism is related to affecting the phosphorylation of key pr...
10074-A4
T9628
10074-A4 is a c-Myc binding compound that associates with c-Myc370–409 and behaves like a “ligand cloud” around a “protein cloud”, with distinct features from th...
KJ Pyr 9
T15665
KJ Pyr 9 is an MYC inhibitor (Kd: 6.5 nM in vitro assay).
MYCMI-6
T12134
MYCMI-6 (NSC-354961) is a potent and selective inhibitor of endogenous MYC:MAX protein interactions,reduces proliferation and induces massive apoptosis in tumor ...
BTYNB
T9033
BTYNB (MDK6620) is an inhibitor of the oncofetal mRNA-binding protein IMP1 (IC50 = 5 μM for IMP1 binding to c-Myc mRNA). MDK6620 downregulates β-TrCP1 mRNA and r...
EN4
T9061
EN4 (EN4 MYC inhibitor) MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It is selective for c-MYC over N-MYC and L-MYC, and inhibits ...
Lusianthridin
TN1892
Lusianthridin is a natural product from Dendrobium venustum. Lusianthridin exhibits anti-migratory property at nontoxic concentrations. Lusianthridin enhances c-...
APTO-253
T10352
APTO-253 (LOR-253) inhibits c-Myc expression, stabilizes G-quadruplex DNA, and induces cell cycle arrest and apoptosis in acute myeloid leukemia cells. APTO-253 ...
ML327
T4252
ML327 is a MYC blocker. ML327 can also de-repress E-cadherin transcription and reverse Epithelial-to-Mesenchymal Transition (EMT).
Mycro 3
T4367
Mycro 3 is potent and selective for c-Myc in whole cell assays.
NY2267
T9093
NY2267 (Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl ester...
10058-F4
T3048
10058-F4 (c-Myc Inhibitor) is a cell-permeable thiazolidinone that specifically inhibits the c-Myc-Max interaction and prevents transactivation of c-Myc target g...
Nicotinamide N-oxide
T0617
Nicotinamide N-oxide (Nicotinamide 1-oxide) is recognized as an in vivo metabolite of nicotinamide which is a precurser of nicotinamide-adenine dinucleotide (NAD...
VPC-70063
T60019
VPC-70063 (Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)-) is an inhibitor of c-Myc-MAX. VPC-70063 exhibits Myc-Max transcriptional activity inh...
Moracin D
TN4581
Moracin C and moracin D, new phytoalexins from diseased mulberry, are antifungal compounds. Moracin may be protective influence in tumor promotion, utilization o...
CBP/p300-IN-2
T10702
CBP/EP300-IN-2 is an inhibitor of CBP/EP300 (IC50s: 1.07 nM and 5.96 nM for CBP/HTRF and Myc) extracted from patent WO2017205538A1 (example 25).
Aaptamine
TN1354
Aaptamine functions as a proteasome inhibitor, it activates p21 promoter in a p53-independent manner.
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