Powder: -20°C for 3 years | In solvent: -80°C for 1 year
(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
5 mg | 在庫あり | ¥ 11,000 | |||
10 mg | 在庫あり | ¥ 15,500 | |||
25 mg | 在庫あり | ¥ 22,500 | |||
50 mg | 在庫あり | ¥ 34,000 | |||
100 mg | 在庫あり | ¥ 54,500 | |||
500 mg | 在庫あり | ¥ 135,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 12,000 |
説明 | (+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1. |
ターゲット&IC50 | PKB AKT:< 0.5 μM, Akt:< 0.5 μM, Akt1:< 0.5 μM, Akt3:< 0.5 μM, PKA:> 5 μM, CDC7:<0.3 nM, PKB AKT2:< 0.5 μM |
別名 | (+)-TBZ, (3R,11bR)-Tetrabenazine, (3R,11bR)-TBZ |
分子量 | 317.42 |
分子式 | C19H27NO3 |
CAS No. | 1026016-83-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 15.0 mg/mL (47.3 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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(+)-Tetrabenazine 1026016-83-0 Membrane transporter/Ion channel Monoamine Transporter (+)-TBZ (3R,11bR)-Tetrabenazine Tetrabenazine (3R,11bR)-TBZ TBZ Inhibitor inhibitor inhibit