Powder: -20°C for 3 years | In solvent: -80°C for 1 year
2-Phenyl-2-(1-piperidinyl)propane (PPP), an analog of phencyclidine
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
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5 mg | 在庫あり | ¥ 11,000 | |||
10 mg | 在庫あり | ¥ 18,500 | |||
25 mg | 在庫あり | ¥ 37,500 | |||
50 mg | 在庫あり | ¥ 57,000 | |||
100 mg | 在庫あり | ¥ 85,500 | |||
200 mg | 在庫あり | ¥ 126,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 11,500 |
説明 | 2-Phenyl-2-(1-piperidinyl)propane (PPP), an analog of phencyclidine |
ターゲット&IC50 | CYP2C9:>300 μM (EC50), CYP2E1:>300 μM (IC50), CYP3A:200 μM (IC50), CYP2C8:>300 μM (IC50), CYP1A2:>300 μM (IC50), CYP2B6:5.1 μM (IC50), CYP2B6:5.6 μM (Ki), CYP2D6:74 μM (IC50), CYP2A6:>300 μM (IC50), CYP2C19:>300 μM (IC50) |
In vivo | 2-Phenyl-2-(1-piperidinyl)propane (PPP) inactivated the 7-(benzyloxy)resorufin O-dealkylation activity of liver microsomes obtained from phenobarbital-induced rats with a K(I) of 11 microM.?The 7-ethoxy-4-(trifluoromethyl)coumarin O-deethylation activity of purified rat liver P450 2B1 and expressed human P450 2B6 was inactivated by PPP in a reconstituted system containing NADPH-cytochrome P450 reductase and lipid[1] |
分子量 | 203.32 |
分子式 | C14H21N |
CAS No. | 92321-29-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 30mg/ml(99.8mM)
You can also refer to dose conversion for different animals. 詳細
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2-Phenyl-2-(1-piperidinyl)propane 92321-29-4 Others 2 Phenyl 2 (1 piperidinyl)propane Reversible inhibit CYPs Cytochrome P450 CYP2B6 CYP3A Inhibitor CYP2D6 2Phenyl2(1piperidinyl)propane inhibitor