Powder: -20°C for 3 years | In solvent: -80°C for 1 year
AMG 9810 is a competitive antagonist of capsaicin activation of the vanilloid receptor 1 (TRPV1) (IC50s = 24.5 and 85.6 nM for human and rat TRPV1, respectively).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
5 mg | 在庫あり | ¥ 10,000 | |||
10 mg | 在庫あり | ¥ 13,000 | |||
25 mg | 在庫あり | ¥ 27,000 | |||
50 mg | 在庫あり | ¥ 49,500 | |||
100 mg | 在庫あり | ¥ 86,500 | |||
500 mg | 在庫あり | ¥ 203,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 11,000 |
説明 | AMG 9810 is a competitive antagonist of capsaicin activation of the vanilloid receptor 1 (TRPV1) (IC50s = 24.5 and 85.6 nM for human and rat TRPV1, respectively). |
ターゲット&IC50 | TRPV1 (rat):85.6 nM, TRPV1 (human):24.5 nM |
In vivo | In a rat model of inflammatory pain induced by intraplantar injection of complete Freund's adjuvant, 30-100 mg/kg AMG 9810 reverses thermal and mechanical hyperalgesia[3]. |
分子量 | 337.41 |
分子式 | C21H23NO3 |
CAS No. | 545395-94-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 33 mg/mL (97.80 mM)
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
AMG9810 545395-94-6 Membrane transporter/Ion channel TRP/TRPV Channel Transient receptor potential channels inhibit Inhibitor AMG-9810 TRP Channel AMG 9810 inhibitor