Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding pA2 values of 4.68. Akuammidine also shows a preference for mu-opioid binding sites with Ki values of 0.6, 2.4 and 8.6 microM at mu-, delta- and kappa-opioid binding sites, respectively.
説明 | Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding pA2 values of 4.68. Akuammidine also shows a preference for mu-opioid binding sites with Ki values of 0.6, 2.4 and 8.6 microM at mu-, delta- and kappa-opioid binding sites, respectively. |
分子量 | 352.43 |
分子式 | C21H24N2O3 |
CAS No. | 642-17-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Akuammigine 642-17-1 Endocrinology/Hormones GPCR/G Protein Neuroscience Adrenergic Receptor Opioid Receptor Inhibitor inhibitor inhibit