Powder: -20°C for 3 years | In solvent: -80°C for 1 year
EP4 Receptor Antagonist 1 is a highly potent and selective competitive prostanoid EP4 receptor antagonist, effective for cancer immunotherapy. It inhibits both human and mouse EP4 receptors with IC50 values of 6.1 nM and 16.2 nM, respectively, while displaying minimal activity (IC50s >10 μM) against human EP1, EP2, and EP3 receptors.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 28,000 | |||
5 mg | 在庫あり | ¥ 72,500 | |||
10 mg | 在庫あり | ¥ 134,500 | |||
25 mg | 在庫あり | お問い合わせ | |||
50 mg | 在庫あり | お問い合わせ |
説明 | EP4 Receptor Antagonist 1 is a highly potent and selective competitive prostanoid EP4 receptor antagonist, effective for cancer immunotherapy. It inhibits both human and mouse EP4 receptors with IC50 values of 6.1 nM and 16.2 nM, respectively, while displaying minimal activity (IC50s >10 μM) against human EP1, EP2, and EP3 receptors. |
ターゲット&IC50 | EP4 receptor (human):6.1 nM , EP4 receptor (mouse):16.2 nM |
分子量 | 458.43 |
分子式 | C23H21F3N4O3 |
CAS No. | 2287259-07-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
EP4 receptor antagonist 1 2287259-07-6 GPCR/G Protein Immunology/Inflammation Prostaglandin Receptor HEK293 EP4 immunotherapy Inhibitor inhibit EP-4 receptor antagonist 1 cells cancer inhibitor