Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約6-8 週間 | ¥ 349,000 |
50 mg | 約6-8 週間 | ¥ 454,500 |
100 mg | 約6-8 週間 | ¥ 574,000 |
説明 | Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM). |
ターゲット&IC50 | mGlu4:79 nM (EC50) |
In vitro | Foliglurax is a highly selective and potent mGlu4 receptor PAM. It has a marked brain-penetrance feature, which might revolutionize the field of mGlu4 receptor drug targeting in CNS disorders [2]. |
別名 | PXT002331 |
分子量 | 421.51 |
分子式 | C23H23N3O3S |
CAS No. | 1883329-51-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 5.2 mg/mL (12.34 mM), Sonication and heating are recommended.
You can also refer to dose conversion for different animals. 詳細
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Foliglurax 1883329-51-8 Neuroscience GluR PXT 002331 PXT-002331 PXT002331 Inhibitor inhibitor inhibit