Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).
パッケージサイズ | 在庫状況 | 単価(税別) | |
---|---|---|---|
1 mg | お問い合わせ | ¥ 25,000 | |
2 mg | お問い合わせ | ¥ 41,000 | |
5 mg | お問い合わせ | ¥ 71,500 | |
10 mg | お問い合わせ | ¥ 111,500 | |
25 mg | お問い合わせ | ¥ 200,500 | |
50 mg | お問い合わせ | ¥ 334,000 | |
100 mg | お問い合わせ | ¥ 455,000 | |
200 mg | お問い合わせ | お問い合わせ | |
500 mg | お問い合わせ | お問い合わせ | |
1 mL * 10 mM (in DMSO) | お問い合わせ | ¥ 77,000 |
説明 | GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM). |
ターゲット&IC50 | GRK2:30 nM, GRK5:7.1 μM |
In vitro | GRKs-IN-1 hydrochloride (Compound 14as) is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine. |
別名 | GRK2-IN-1 hydrochloride |
分子量 | 488.94 |
分子式 | C24H26ClFN4O4 |
CAS No. | T13714L |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL (511.31 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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GRK2-IN-1 hydrochloride (2055990-90-2 free base) T13714L GPCR/G Protein GRK GRK2-IN-1 Hydrochloride 2055990-90-2 GRK-2-IN-1 hydrochloride (2055990-90-2 free base) GRK2IN1 hydrochloride (2055990902 free base) GRK2-IN-1 hydrochloride 2055990-90-2 free base GRK2 IN 1 hydrochloride (2055990 90 2 free base) Inhibitor inhibitor inhibit