Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GSK270822A is a selective ROCK1 inhibitor. GSK270822A exhibits IC50 of 9nM, 1100nM, 1550nM for ROCK1, RSK1, p70S6K, respectively.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 91,500 |
5 mg | 在庫あり | ¥ 223,000 |
10 mg | 在庫あり | ¥ 296,000 |
25 mg | 在庫あり | ¥ 447,500 |
50 mg | 在庫あり | ¥ 601,500 |
100 mg | 在庫あり | ¥ 810,500 |
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 228,500 |
説明 | GSK270822A is a selective ROCK1 inhibitor. GSK270822A exhibits IC50 of 9nM, 1100nM, 1550nM for ROCK1, RSK1, p70S6K, respectively. |
In vitro | GSK270822A inhibits rat aortic ring dilation with IC50 of 76nM[1]. |
別名 | GSK 270822A, GSK-270822A |
分子量 | 396.44 |
分子式 | C24H20N4O2 |
CAS No. | 864082-23-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (126.12 mM)
You can also refer to dose conversion for different animals. 詳細
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GSK270822A 864082-23-5 GPCR/G Protein GRK GSK 270822A GSK-270822A Inhibitor inhibitor inhibit