store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Glutaminase-IN-1 (CB839 derivative), a novel 1,3,4-selenodiazepine renal-type glutaminase (KGA) variant inhibitor, showed antitumor activity in an aggressive H22 hepatocellular carcinoma xenograft model.
ターゲット&IC50 | A549 cells:17 nM, KGA:1 nM, HCT116 cells:9 nM, Caki-1 cells:19 nM, H2:6.78 μM |
別名 | CB839 derivative |
分子量 | 618.47 |
分子式 | C26H24F3N7O3Se |
CAS No. | 2247127-79-1 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (161.69 mM), Sonication is recommended.
H2O: 1 mg/mL (1.61 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Glutaminase-IN-1 2247127-79-1 Metabolism transporter GlutaminaseIN1 CB839 derivative Glutaminase IN 1 Inhibitor inhibitor inhibit