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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T22714 | Decynium 22 | Others | |
Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor | |||
T9558 | KL-11743 | transporter | |
KL-11743 specifically blocks glucose metabolism, triggering an acute collapse in NADH pools and a striking accumulation of aspartate, indicating a dramatic shift toward oxidative phosphorylation in the mitochondria. | |||
T3713 | BAY-876 | transporter | |
BAY-876 is an orally active and selective inhibitor of glucose transporter 1 (GLUT1, IC50= 2 nM). BAY-876 exhibits >130-fold more selective for GLUT1 than GLUT2, GLUT3, and GLUT4. BAY-876 also inhibits glycolytic metabol... | |||
T7147 | Valbenazine | NBI-98854 | Monoamine Transporter |
Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia. | |||
T23070 | Nisoxetine hydrochloride | Sodium Channel , Monoamine Transporter , Norepinephrine | |
Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitor | |||
T9347 | EAAT2 activator 1 | 3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine | transporter |
EAAT2 activator 1 (3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine) is a thiopyridazine derivative that has been found to increase EAAT2 protein levels in astrocytes. | |||
T39429 | AHN 1-055 hydrochloride | 3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride | Dopamine Receptor |
AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM). | |||
T11087 | DOV-216,303 Free Base | DOV-216303 | Dopamine Receptor , Serotonin Transporter , Norepinephrine |
T7018 | WZB117 | transporter | |
WZB117 is a Glucose Transporter 1 (GLUT1) inhibitor. when IC50 of WZB117 approximate 10 μM, it inhibits lung cancer A549 cells and breast cancer MCF7 cells proliferation. | |||
T10758L | Centanafadine hydrochloride | EB-1020 hydrochloride | Dopamine Receptor , Serotonin Transporter , Adrenergic Receptor , Norepinephrine |
Centanafadine hydrochloride (EB-1020 hydrochloride) is a dual inhibitor of norepinephrine (NE)/dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 83 nM for human NE, DA, and serotonin... | |||
T12232 | Nitroxazepine | CIBA 2330Go | Serotonin Transporter |
Nitroxazepine (CIBA 2330Go) is a serotonin-norepinephrine reuptake inhibitor, and treatment depression. Nitroxazepine is a tricyclic antidepressant (TCA) for the research of depression | |||
T1768 | 7ACC2 | Mitochondrial Metabolism , Monocarboxylate transporter | |
7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for [14C]-lactate influx; new antitumor treatment targeting lactate transport in Y cells. | |||
T5208 | BAY-8002 | BAY8002,BAY 8002 | Monocarboxylate transporter |
BAY-8002 is a potent dual MCT1/2 inhibitor (IC50 values are 3, 8, and 12 nM at rat (C6), human (DLD-1) and mouse (4T1) MCT1 respectively). | |||
T8708 | Paroxetine | Serotonin Transporter | |
Paroxetine is a inhibitor of serotonin uptake that is effective in the treatment of depression. | |||
T3210 | AZD3965 | AZD 3965,AZD-3965 | Monocarboxylate transporter |
AZD3965 (AZD-3965) is a selective inhibitor of monocarboxylate transporter 1 (MCT1). | |||
T3526 | Dasotraline hydrochloride | SEP-225289 hydrochloride | Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Norepinephrine |
Dasotraline hydrochloride (SEP-225289 hydrochloride) (SEP-225289 hydrochloride) is a triple reuptake inhibitor that inhibits dopamine, norepinephrine, and serotonin transporters with IC50 values of 4, 6, and 11 nM, respe... | |||
T15411 | GPNA hydrochloride | Apoptosis , Others | |
GPNA hydrochloride is specific glutamine (Gln) transporter ASCT2(SLC1A5) inhibitor. GPNA reversibly induces apoptosis in A549 cells. GPNA hydrochloride is a well-known substrate of the enzyme γ-glutamyltransferase (GGT).... | |||
T14316 | AR-C155858 | Monocarboxylate transporter | |
AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM). | |||
T11064 | DMT1 blocker 2 | Others | |
DMT1 blocker 2, compound 12f, is a direct inhibitor of divalent metal transporter 1 (DMT1) with an IC50 hydrogen peroxide value of 0.83, which is expected to block iron uptake by intestinal epithelial cells in vivo. | |||
T2363 | STF-31 | transporter , Autophagy | |
STF-31 is an inhibitor of glucose transporter 1 (GLUT1) with IC50 of 1 μM. | |||
T7341 | Diclofensine | Ro 8-4650 | Dopamine Receptor , Monoamine Transporter |
Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine. | |||
T0322 | Fipexide | Dopamine Receptor , AChR | |
Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983. It was served as a nootropic drug in France and Italy, mainly for the therapy of senile dementia, but is... | |||
T6414 | Bisacodyl | Fenilaxan,Dulcolax,Brocalax | Others |
Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation. | |||
T8732 | CTPI-2 | Others , Mitochondrial Metabolism | |
CTPI-2 is an inhibitor of mitochondrial citrate carrier SLC25A1 with(KD : 3.5 μM). CTPI-2 inhibits glycolysis, PPARγ, and its downstream target the glucose transporter GLUT4. CTPI-2 exhibits anti-tumor activity.CTPI-2 ha... | |||
T7061 | Duloxetine | Serotonin Transporter | |
Duloxetine is an inhibitor of serotonin-norepinephrine reuptake(Ki of 4.6 nM),with treatment of major depressive disorder and generalized anxiety disorder. | |||
T3994 | Verinurad | RDEA3170 | OAT |
Verinurad (RDEA3170) (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for the treatment of gout and hyperuricemia. | |||
T5345 | V-9302 | Others | |
V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 (IC50: 9.6 uM). | |||
T2092 | Amitifadine hydrochloride | DOV-21947 hydrochloride,EB-1010 hydrochloride | Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Norepinephrine |
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI). | |||
T4182 | Lavendustin B | Tyrosinase , transporter , HIV Protease | |
Lavendustin B is a Tyrosine Kinase Inhibitor and an inhibitor of HIV-1 integrase (IN) interaction with its cognate cellular cofactor, lens epithelium-derived growth factor (LEDGF/p75). | |||
T0450 | Fluoxetine | LY-110140 | 5-HT Receptor , Serotonin Transporter , MRP , Autophagy |
Fluoxetine (LY-110140) is a highly specific serotonin uptake inhibitor and selective 5-hydroxytryptamine (5-HT) reuptake inhibitor. Fluoxetine has antidepressant activity. | |||
T15728 | LDN-212320 | LDN-0212320,LDN/OSU-0212320,OSU-0212320 | transporter |
LDN-212320 (OSU-0212320) is a glutamate transporter EAAT2 activator. It also enhances EAAT2 levels by > 6 fold at concentrations < 5 μM after 24 h. | |||
T20545 | Benzarone | Benzarona,Vasoc,Venagil,Benzaronum | OAT |
Benzarone (Benzarona) is a potent inhibitor of human uric acid transporter 1 (URAT1, IC50 = 2.8 μM in oocyte). Benzarone lowers the level of uric acid serum. | |||
T6875 | Lesinurad | RDEA594 | OAT |
Lesinurad (RDEA594) is a selective inhibitor of uric acid reabsorption which is used in combination with other agents in the therapy of gout. Lesinurad has had a limited clinical use but has not been associated with seru... | |||
T6697 | TCID | UCH-L3 Inhibitor | DUB |
TCID (UCH-L3 Inhibitor)(IC50=0.6 μM) is a DUB inhibitor of ubiquitin C-terminal hydrolase L3. It has the 125-fold selectivity to L1. | |||
T0719 | Tetrabenazine | Xenazine,Ro 1-9569 | Others , Dopamine Receptor , Monoamine Transporter |
Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders. Tetrabenazine blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high... | |||
T8551 | Nitrobenzylthioinosine | NBMPR | AChR , Adenosine Receptor |
Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity. | |||
T0413 | Cinromide | trans-3-Bromo-N-ethylcinnamamide | Others |
Cinromide (trans-3-Bromo-N-ethylcinnamamide) is used as a novel anticonvulsant agent. | |||
T0991 | Desipramine hydrochloride | NSC-114901,Desmethylimipramine,JB-8181,EX-4355,Norimipramine,G-35020 | Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Adrenergic Receptor |
Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervous system (CNS), Desipramine hydrochloride blocks the re-upt... | |||
T22453 | Venlafaxine | Wy 45030 | Serotonin Transporter |
Venlafaxine (Wy 45030), an arylalkanolamine serotonin-norepinephrine reuptake inhibitor (SNRI), is used to treat major generalised anxiety disorder (GAD), depressive disorder (MDD), panic disorder and social phobia. | |||
T1189 | Milnacipran hydrochloride | Milnacipran HCl,Savella,Dalcipran | Serotonin Transporter , Norepinephrine |
Milnacipran hydrochloride (Savella) is a serotonin and norepinephrine reuptake inhibitor used to treat major depressive disorders. Milnacipran hydrochloride is an enantiomer of milnacipran, which is used to treat fibromy... | |||
T2594 | Dextromilnacipran | Levomilnacipran | Serotonin Transporter , Norepinephrine |
Dextromilnacipran (Levomilnacipran) is a selective serotonin and norepinephrine reuptake inhibitor. | |||
T1871 | GBR 12935 dihydrochloride | GBR12935,GBR-12935,GBR 12935 | Dopamine Receptor |
GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels. | |||
T0766 | Promazine hydrochloride | Romtiazin hydrochloride,Sinophenin hydrochloride | Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , AChR |
Promazine hydrochloride (Romtiazin hydrochloride) is a phenothiazine with actions similar to CHLORPROMAZINE but with less antipsychotic activity. It is primarily used in short-term treatment of disturbed behavior and as ... | |||
T2556 | Nandrolone decanoate | 19-Nortestosterone decanoate | Others , HIV Protease |
Nandrolone decanoate (19-Nortestosterone decanoate) is the decanoate salt form of nandrolone, an anabolic steroid analog of testosterone with androgenic, anabolic, and erythropoietin stimulating effects. Nandrolone enter... | |||
T1993 | J-147 | J147 | Epigenetic Reader Domain , Dopamine Receptor , Monoamine Oxidase |
J-147 is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging. It is a curcumin derivative and a potent neurogenic and neuroprotective drug candidate... | |||
T8616 | Fasentin | N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide | transporter |
Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) is an inhibitor of GluT1. | |||
T7460 | α-Cyano-4-hydroxycinnamic acid | α-Cyano-4-hydroxycinnamic acid(α-CHCA) | Monocarboxylate transporter |
α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvate transport in rat heart mitochondria (IC50 : 1.5 μM). | |||
T1580 | Desvenlafaxine | WY 45233 Succinate,O-Desmethylvenlafaxine | 5-HT Receptor , Serotonin Transporter , Norepinephrine |
Desvenlafaxine (O-Desmethylvenlafaxine) is a cyclohexanol and phenol derivative and metabolite of venlafaxine that functions as a serotonin and noradrenaline reuptake inhibitor (SNRI) and is used as an antidepressive age... | |||
T2227 | Hemicholinium 3 | Hemicholinium-3,Hemicholine | Others , AChE |
Hemicholinium 3 is a potent and selective choline uptake blocker. | |||
T7940 | Milnacipran ((1S-cis) hydrochloride) | Levomilnacipran Hydrochloride | Serotonin Transporter |
Milnacipran (1S-cis) hydrochloride (Levomilnacipran Hydrochloride) is a serotonin-norepinephrine reuptake inhibitor (SNRI), treatment of fibromyalgia. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
TN6552 | 5,7-Dimethoxyluteolin | Dopamine Receptor | |
5,7-Dimethoxyluteolin is a natural product from Hovenia acerba. 5,7-Dimethoxyluteolin is a dopamine transporter (DAT) activator with an EC50 of 3.417 μM. | |||
T0791 | Reserpine | Serpalan,Serpasil,Serpivite | Others , Potassium Channel , MRP , Monoamine Transporter , Autophagy |
Reserpine (Serpalan) is an alkaloid found in the roots of Rauwolfia serpentina and R. vomitoria. Reserpine inhibits the uptake of norepinephrine into storage vesicles resulting in depletion of catecholamines and serotoni... | |||
TN2252 | Syrosingopine | Dopamine Receptor | |
Syrosingopine has selective depleting effect on brain amines is potentiated by combined treatment with disulfiram or fusaric acid, a dopamine beta-hydroxylase inhibitor. | |||
TN1118 | Tormentic acid | Immunology/Inflammation related | |
Tormentic acid is a natural product. It has anticancer, anti-inflammatory, anti-atherogenic , anti-allodynic, and hepatoprotective properties, | |||
T4S1545 | Licarin B | (-)-Licarin B,Licarine B | transporter , Antibacterial , PPAR |
1.(-)-Licarin B (Licarine B) has anti-mycobacterial activity. | |||
T7521 | Azaphen | Pipofezin hydrochloride,Pipofezine hydrochloride,Azafen | 5-HT Receptor , Serotonin Transporter |
Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity. | |||
T1317 | Cinchonidine | α-Quinidine,L-Cinchonidine | 5-HT Receptor , Serotonin Transporter , Parasite |
Cinchonidine (L-Cinchonidine) is an alkaloid extracted from Cinchona officinalis. It is a pseudo-enantiomer and stereoisomer of cinchonine. | |||
T3S0364 | L-Arginine | L-Arg,(S)-(+)-Arginine | IL Receptor , Endogenous Metabolite , NO Synthase |
1. L-Arginine (L-Arg) exhibits anti-atherosclerotic effect. 2. L-Arginine and soy enriched diet are effective in prevention of osteoporosis associated with diabetes mellitus. 3. Exogenous L-Arginine could enhance neonate... | |||
T2203 | D-Carnitine hydrochloride | (S)-Carnitine Hydrochloride,L-Carnitine hydrochloride | Others , Endogenous Metabolite |
D-Carnitine hydrochloride ((S)-Carnitine Hydrochloride) is a constituent of striated muscle and liver. It is used therapeutically to stimulate gastric and pancreatic secretions and in the treatment of hyperlipoproteinemi... | |||
T0185 | Escitalopram | Seroplex,S-(+)-Citalopram,(S)-Citalopram | Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Adrenergic Receptor , AChR , Norepinephrine , Histamine Receptor |
Escitalopram (Seroplex) is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol uptake in alcoholics and is used in depressed patien... | |||
T2924 | Phloretin | Dihydronaringenin,NSC 407292,RJC 02792 | SGLT , transporter , Endogenous Metabolite |
Phloretin (NSC-407292) is a well-known inhibitor of eukaryotic urea transporters, blocks VacA-mediated urea and ion transport. Phloretin is a dihydrochalcone, a type of natural phenols. It can be found in apple tree leav... | |||
T6S0117 | Avicularin | Fenicularin | ERK |
Avicularin (Fenicularin) has anti-allergic, anti-inflammatory, hepatoprotective, antioxidant, anti-tumor and other activities. It ameliorates human hepatocellular carcinoma by modulating the activities of NF-κB(p65), COX... | |||
TN1033 | Sennidin A | HCV Protease , transporter , Akt , PI3K | |
Sennidin A, has two hydroxyanthraquinone-like moieties, exerts inhibition on NS3 helicase with IC50 values of 0.8 μM. | |||
TN1034 | Sennidin B | HCV Protease , transporter , Akt , PI3K | |
Sennidin B stimulates glucose incorporation in rat adipocytes. | |||
T2755 | Rhoifolin | Apigenin-7-O-rhamnoglucoside,Apigenin 7-O-neohesperidoside,Rhoifoloside | Others , p38 MAPK , NF-κB , transporter , IGF-1R , Autophagy |
Rhoifolin (Apigenin 7-O-neohesperidoside) is extracted from Turpinia arguya Seem dried leaves. | |||
T19866 | Indican | NSC-87517,3-Indoxyl-beta-D-glucopyranoside,NSC 87517,NSC87517,Indoxyl-β-D-glucoside | OAT , MRP |
Indican (Indoxyl-β-D-glucoside) is a natural protective compound that is used to protect the liver. | |||
T4702 | (3-Carboxypropyl)trimethylammonium chloride | γ-Butyrobetaine hydrochloride,(3-Carboxypropyl)trimethylammonium chlor | Endogenous Metabolite |
(3-Carboxypropyl)trimethylammonium chloride ((3-Carboxypropyl)trimethylammonium chlor) is a synthetic carnitine related compound used as a transporter substrate in the cloning and sequencing of human carnitine transporte... | |||
TN5118 | Taxol C | P-gp | |
Taxol C can reduce interaction with the P-glycoprotein transporter that may allow for increased permeation of taxanes into the brain. | |||
T4912 | Jatrorrhizine chloride | Yatrorhizine chloride,Neprotine chloride | Others , 5-HT Receptor , OCT , Antibacterial , AChE |
Jatrorrhizine chloride (Neprotine chloride) is a potent and orally active uptake-2 transporter inhibitor. It exhibits a critical neuroprotective role in H2O2-induced apoptosis via inhibition of the MAPK pathway in HT22 h... | |||
T13655 | DL-Norepinephrine hydrochloride | Lys,DL-lysine | Adrenergic Receptor |
DL-Norepinephrine hydrochloride (DL-lysine) is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400 μM. | |||
T6975 | Sarcosine | Sarcosinic acid,Methylaminoacetic acid,Sarcosin,Methylglycine,N-Methylaminoacetic acid,N-methylglycine | Others , GlyT , Endogenous Metabolite |
Sarcosine (Methylglycine) is a competitive inhibitor of the type I glycine transporter (GlyT1) and an N-methyl-D-aspartate receptor (NMDAR) co-agonist. | |||
T1153 | Trimethoprim | NIH 204,BW 56-72,NSC-106568 | DHFR , DNA/RNA Synthesis , Antifolate , Antibacterial , Antibiotic |
Trimethoprim (NSC-106568) is a Dihydrofolate Reductase Inhibitor Antibacterial. The mechanism of action of trimethoprim is as a Dihydrofolate Reductase Inhibitor, and Cytochrome P450 2C8 Inhibitor, and Organic Cation Tra... | |||
T4S0779 | D-tetrahydropalmatine | Others , Dopamine Receptor | |
D-Tetrahydropalmatine is a organic cation transporter 1 (OCT1) inhibitor, it can obviously inhibit the uptake of monocrotaline (MCT) in MDCK-hOCT1 cells and isolate rat primary hepatocytes, and attenuate the viability re... | |||
T3933 | Jatrorrhizine | Yatrorizine,neprotin | MAO , 5-HT Receptor , Antibacterial , AChE |
Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species. It was found to have antimicrobial and antifungal activity. It binds and noncompetitively inhibits mo... | |||
T19772 | Mesembrenone | (+)-Mesembrenone | |
Mesembrenone is a selective the serotonin transporter (SERT) inhibitor. Mesembrenone is the main alkaloid of Sceletium tortuosum. | |||
T80013 | Arecaidine hydrobromide | GABA Receptor | |
Arecaidine hydrobromide, a pyridine alkaloid, functions as a potent GABA uptake inhibitor and acts as a substrate for the H+-coupled amino acid transporter 1 (PAT1, SLC36A1), where it competitively inhibits L-proline upt... | |||
T72961 | Falcarindiol | 法卡林二醇 | |
Falcarindiol, an orally active polyacetylenic oxylipin, not only activates PPARγ, enhancing ABCA1 expression—a cholesterol transporter—but also induces apoptosis and autophagy. This compound exhibits anti-inflammatory, a... | |||
T72645 | Norbatzelladine L | ||
Norbatzelladine L, an inhibitor of both the catalytic and functional activities of the Pdr5p transporter, suppresses Pdr5p ATPase activity with an IC50 of 3.8 µM. Additionally, it exhibits antifungal, antiparasitic, anti... | |||
T72172 | 4,6-O-Ethylidene-α-D-glucose | Ethylidene-glucose | |
4,6-O-Ethylidene-α-D-glucose (Ethylidene-glucose), a derivative of glucose, serves as a competitive inhibitor for the exofacial binding site of glucose transporter 1 (GLUT1), exhibiting a Ki of 12 mM against wild-type 2-... | |||
T73857 | Mesembrine | ||
Mesembrine ((+)-Mesembrine), a primary alkaloid distinguished by its aryloctahydroindole structure, acts as a potent 5-HT transporter inhibitor with an inhibition constant (K i) of 1.4 nM. Additionally, it demonstrates i... | |||
T80014 | Guvacine hydrobromide | GABA Receptor | |
Guvacine hydrobromide, an alkaloid derived from the Areca catechu nut, serves as a potent inhibitor of GABA (GABA uptakp) uptake. It effectively inhibits rat GABA transporter isoforms GAT-1, GAT-2, and GAT-3, with respec... | |||
T37810 | 6',7'-Epoxybergamottin | ||
6'7'-Epoxybergamottin is a furanocoumarin found in grapefruit. It is a potent inhibitor of the cytochrome P450 (CYP) isoform CYP3A4 with an IC50 value of 0.30 ppm in a cell-free assay, 0.33 μM in HL7 human liver cells, a... | |||
T19290 | DL-Lysine | (±)-2,6-Diaminocaproic acid | Others |
DL-Lysine (Lysine) is an α-amino acid that is used in the biosynthesis of proteins. | |||
T75436 | Jatrorrhizine hydroxide | ||
Jatrorrhizine hydroxide, an alkaloid derived from Coptis chinensis, exhibits a range of biological activities including neuroprotective, antimicrobial, antiplasmodial, and antioxidant properties [1]. It acts as a potent ... |
カタログ番号 | 製品名 | Species | Expression System |
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TMPY-05650 | FCGRT & B2M Heterodimer Protein, Cynomolgus, Recombinant (His & Avi), Biotinylated | Cynomolgus | HEK293 |
FCGRT & B2M Heterodimer Protein, Cynomolgus, Recombinant (His & Avi), Biotinylated is expressed in HEK293 cells. | |||
TMPY-02829 | FCGRT & B2M Heterodimer Protein, Rat, Recombinant (His) | Rat | HEK293 |
FCGRT & B2M Heterodimer Protein, Rat, Recombinant (His) is expressed in HEK293 with His tag. The predicted molecular weight is 44 kDa. Accession number: P13599&P07151 | |||
TMPY-02830 | FCGRT & B2M Heterodimer Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 |
FCGRT & B2M Heterodimer Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 with His tag. The predicted molecular weight is 43.5 kDa. Accession number: Q8SPV9&Q8SPW0 | |||
TMPY-02811 | FCGRT & B2M Heterodimer Protein, Mouse, Recombinant (His) | Mouse | HEK293 |
FCGRT & B2M Heterodimer Protein, Mouse, Recombinant (His) is expressed in HEK293 with His tag. The predicted molecular weight is 43.5 kDa. Accession number: Q61559&P01887 | |||
TMPY-02082 | FCGRT & B2M Heterodimer Protein, Human, Recombinant (His) | Human | HEK293 |
FCGRT & B2M Heterodimer Protein, Human, Recombinant (His) is expressed in HEK293 cells. | |||
TMPY-05539 | FCGRT & B2M Heterodimer Protein, Human, Recombinant (His), Biotinylated | Human | HEK293 |
FCGRT & B2M Heterodimer Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 cells. | |||
TMPY-01938 | CD98 Protein, Human, Recombinant (His) | Human | HEK293 |
4F2 cell-surface antigen heavy chain, also known as 4F2 heavy chain antigen, Lymphocyte activation antigen 4F2 large subunit, CD98, SLC3A2 and MDU1, is a single-pass type I I membrane protein that belongs to the SLC3A tr... | |||
TMPY-02209 | CUTC Protein, Human, Recombinant (His) | Human | E. coli |
Copper homeostasis protein cutC homolog, also known as CGI-32 and CUTC, is a cytoplasm and nucleus protein which belongs to theCutC family. CUTC may play a role in copper homeostasis. It can bind one Cu1+per subunit. ... | |||
TMPY-02358 | CD98 Protein, Mouse, Recombinant (His) | Mouse | HEK293 |
4F2 cell-surface antigen heavy chain, also known as 4F2 heavy chain antigen, Lymphocyte activation antigen 4F2 large subunit, CD98, SLC3A2 and MDU1, is a single-pass type I I membrane protein that belongs to the SLC3A tr... | |||
TMPY-05149 | FCGRT & B2M Heterodimer Protein, Cynomolgus, Recombinant (His), Biotinylated | Cynomolgus | HEK293 |
FCGRT & B2M Heterodimer Protein, Cynomolgus, Recombinant (His), Biotinylated is expressed in HEK293 with His tag. The predicted molecular weight is 43.5 kDa. Accession number: Q8SPV9&Q8SPW0 | |||
TMPY-05148 | FCGRT & B2M Heterodimer Protein, Rat, Recombinant (His), Biotinylated | Rat | HEK293 |
FCGRT & B2M Heterodimer Protein, Rat, Recombinant (His), Biotinylated is expressed in HEK293 with His tag. The predicted molecular weight is 44 kDa. Accession number: P13599&P07151 | |||
TMPY-05147 | FCGRT & B2M Heterodimer Protein, Mouse, Recombinant (His), Biotinylated | Mouse | HEK293 |
FCGRT & B2M Heterodimer Protein, Mouse, Recombinant (His), Biotinylated is expressed in HEK293 with His tag. The predicted molecular weight is 44.2 kDa. Accession number: Q61559&P01887 | |||
TMPY-03857 | MMGT1 Protein, Human, Recombinant (His) | Human | HEK293 |
MMGT1 (Membrane Magnesium Transporter 1, also known as EMC5 and TMEM32) is a Protein Coding gene. 2 alternatively spliced human isoforms have been reported. The encoded protein belongs to the membrane magnesium transport... | |||
TMPY-05649 | FCGRT & B2M Heterodimer Protein, Mouse, Recombinant (His & Avi), Biotinylated | Mouse | HEK293 |
FCGRT & B2M Heterodimer Protein, Mouse, Recombinant (His & Avi), Biotinylated is expressed in HEK293 with His and AVI tag. The predicted molecular weight is 46 kDa. Accession number: Q61559 | |||
TMPY-05448 | FCGRT & B2M Heterodimer Protein, Human, Recombinant (His & Avi), Biotinylated | Human | HEK293 |
FCGRT & B2M Heterodimer Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 with His and AVI tag. The predicted molecular weight is 45.3 kDa. Accession number: NP_004098.1&NP_004039.1 | |||
TMPY-05036 | FCGRT & B2M Heterodimer Protein, Human, Recombinant (His & Avi) | Human | HEK293 |
FCGRT & B2M Heterodimer Protein, Human, Recombinant (His & Avi) is expressed in HEK293 with His and AVI tag. The predicted molecular weight is 45.3 kDa. Accession number: NP_004098.1&NP_004039.1 | |||
TMPY-04631 | CD98 Protein, Rat, Recombinant (hFc) | Rat | HEK293 |
4F2 cell-surface antigen heavy chain, also known as 4F2 heavy chain antigen, Lymphocyte activation antigen 4F2 large subunit, CD98, SLC3A2 and MDU1, is a single-pass type I I membrane protein that belongs to the SLC3A tr... | |||
TMPY-03307 | CD98 Protein, Rat, Recombinant (His) | Rat | HEK293 |
4F2 cell-surface antigen heavy chain, also known as 4F2 heavy chain antigen, Lymphocyte activation antigen 4F2 large subunit, CD98, SLC3A2 and MDU1, is a single-pass type I I membrane protein that belongs to the SLC3A tr... | |||
TMPH-01711 | ABCC1 Protein, Human, Recombinant (His) | Human | E. coli |
Mediates export of organic anions and drugs from the cytoplasm. Mediates ATP-dependent transport of glutathione and glutathione conjugates, leukotriene C4, estradiol-17-beta-o-glucuronide, methotrexate, antiviral drugs a... | |||
TMPY-01118 | SLC27A4/FATP4 Protein, Human, Recombinant (His) | Human | HEK293 |
SLC27A4/ATG4B complex might act as a new potential therapeutic target of lung tumor chemotherapy. The solute carrier 27A (SLC27A) gene family encodes fatty acid transport proteins (FATPs) and includes 6 members. Autism s... | |||
TMPJ-00583 | CDH17 Protein, Human, Recombinant (His) | Human | Human Cells |
Cadherin-17 is a single-pass type I membrane protein that belongs to the cadherin superfamily. Cadherin-17 consists of one extracellular region containing seven cadherin domains and one transmembrane region but it lacks ... | |||
TMPY-06611 | CD98 Protein, Human, Recombinant (His), Biotinylated | Human | HEK293 |
4F2 cell-surface antigen heavy chain, also known as 4F2 heavy chain antigen, Lymphocyte activation antigen 4F2 large subunit, CD98, SLC3A2 and MDU1, is a single-pass type I I membrane protein that belongs to the SLC3A tr... | |||
TMPH-00981 | ABCB1 Protein, Human, Recombinant (His) | Human | E. coli |
ABCB1 Protein, Human, Recombinant (His) is expressed in E. coli. | |||
TMPH-00206 | Pertactin autotransporter Protein, Bordetella pertussis, Recombinant (His & SUMO) | Bordetella pertussis | E. coli |
Agglutinogen that binds to eukaryotic cells; a process mediated by the R-G-D sequence. Pertactin may have a role in bacterial adhesion, and thus play a role in virulence. May contribute to the disease state of whooping c... | |||
TMPY-03120 | Prostaglandin D2 Synthase Protein, Human, Recombinant (His) | Human | HEK293 |
PTGDS, also known as L-PGDS, belongs to the calycin superfamily, lipocalin family. Lipocalins share limited regions of sequence homology and a common tertiary structure architecture. They transport small hydrophobic mole... | |||
TMPY-05047 | CD44 Protein, Mouse, Recombinant (His) | Mouse | HEK293 |
CD44 is a type I transmembrane protein and a member of the cartilage link protein family. It is involved in cell-cell and cell-matrix interactions and signal transduction. Several CD44 ligands have been identified. The m... | |||
TMPY-02033 | CD44 Protein, Human, Recombinant (His) | Human | HEK293 |
CD44 is a type I transmembrane protein and a member of the cartilage link protein family. It is involved in cell-cell and cell-matrix interactions and signal transduction. Several CD44 ligands have been identified. The m... | |||
TMPY-01146 | Insulin Receptor Protein, Human, Recombinant (long isoform, His) | Human | HEK293 |
INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to the protein kinase superfamily and exists as a tetramer consisting of two alpha subunits and two beta... | |||
TMPY-05352 | Cadherin 17/CDH17 Protein, Cynomolgus, Recombinant (hFc) | Cynomolgus | HEK293 |
Cadherin-17 or LI-cadherin is a member of the cadherin superfamily, genes encoding calcium-dependent, membrane-associated glycoproteins. Cadherin-17/LI-cadherin is a cadherin-like protein consisting of an extracellular r... | |||
TMPY-01912 | Cadherin 17/CDH17 Protein, Human, Recombinant (His) | Human | HEK293 |
Cadherin-17 or LI-cadherin is a member of the cadherin superfamily, genes encoding calcium-dependent, membrane-associated glycoproteins. Cadherin-17/LI-cadherin is a cadherin-like protein consisting of an extracellular r... | |||
TMPY-02919 | Cadherin 17/CDH17 Protein, Rat, Recombinant (His) | Rat | HEK293 |
Cadherin-17 or LI-cadherin is a member of the cadherin superfamily, genes encoding calcium-dependent, membrane-associated glycoproteins. Cadherin-17/LI-cadherin is a cadherin-like protein consisting of an extracellular r... | |||
TMPH-02333 | SLC25A19 Protein, Human, Recombinant (His) | Human | in vitro E. coli expression system |
Mitochondrial transporter mediating uptake of thiamine pyrophosphate (ThPP) into mitochondria. | |||
TMPH-02324 | SLC39A6 Protein, Human, Recombinant (His) | Human | Baculovirus |
May act as a zinc-influx transporter. | |||
TMPH-03414 | RT0041 Protein, Rickettsia typhi, Recombinant (His & Myc) | Rickettsia typhi | E. coli |
Could be part of an ABC transporter complex. | |||
TMPH-03591 | PsaA Protein, S. pneumoniae, Recombinant (His & Myc) | Streptococcus pneumoniae | E. coli |
Part of an ABC transporter complex involved in manganese import. | |||
TMPH-00628 | GltI/YbeJ Protein, E. coli, Recombinant (His & SUMO) | E. coli | E. coli |
Part of the ABC transporter complex GltIJKL involved in glutamate and aspartate uptake. Binds to both glutamate and aspartate. | |||
TMPH-00652 | MMBP Protein, E. coli, Recombinant (His & Myc) | E. coli | E. coli |
Part of the ABC transporter complex MalEFGK involved in maltose/maltodextrin import. Binds maltose and higher maltodextrins such as maltotriose. | |||
TMPH-02123 | SLC2A9 Protein, Human, Recombinant (His) | Human | in vitro E. coli expression system |
Urate transporter, which may play a role in the urate reabsorption by proximal tubules. Does not transport glucose, fructose or galactose. | |||
TMPH-02177 | Tapasin Protein, Human, Recombinant (His & Myc) | Human | E. coli |
Involved in the association of MHC class I with transporter associated with antigen processing (TAP) and in the assembly of MHC class I with peptide (peptide loading). | |||
TMPH-00787 | BtuD Protein, Halobacterium salinarum, Recombinant | Halobacterium salinarum | E. coli |
Required for corrinoid utilization. Probably part of the ABC transporter complex BtuCDF involved in cobalamin (vitamin B12) import. Probably responsible for energy coupling to the transport system. | |||
TMPH-00786 | BtuD Protein, Halobacterium salinarum, Recombinant (His) | Halobacterium salinarum | E. coli |
Required for corrinoid utilization. Probably part of the ABC transporter complex BtuCDF involved in cobalamin (vitamin B12) import. Probably responsible for energy coupling to the transport system. | |||
TMPH-02554 | BCAT2 Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
Catalyzes the first reaction in the catabolism of the essential branched chain amino acids leucine, isoleucine, and valine. May also function as a transporter of branched chain alpha-keto acids. | |||
TMPH-02979 | SLC30A8 Protein, Mouse, Recombinant (His) | Mouse | in vitro E. coli expression system |
Facilitates the accumulation of zinc from the cytoplasm into intracellular vesicles, being a zinc-efflux transporter. May be a major component for providing zinc to insulin maturation and/or storage processes in insulin-... | |||
TMPH-02323 | SLC30A8 Protein, Human, Recombinant (His) | Human | in vitro E. coli expression system |
Facilitates the accumulation of zinc from the cytoplasm into intracellular vesicles, being a zinc-efflux transporter. May be a major component for providing zinc to insulin maturation and/or storage processes in insulin-... | |||
TMPH-01696 | SLC16A4 Protein, Human, Recombinant (His) | Human | E. coli |
Proton-linked monocarboxylate transporter. Catalyzes the rapid transport across the plasma membrane of many monocarboxylates such as lactate, pyruvate, branched-chain oxo acids derived from leucine, valine and isoleucine... | |||
TMPH-01390 | G6PC Protein, Human, Recombinant (His & SUMO) | Human | E. coli |
Hydrolyzes glucose-6-phosphate to glucose in the endoplasmic reticulum. Forms with the glucose-6-phosphate transporter (SLC37A4/G6PT) the complex responsible for glucose production in the terminal step of glycogenolysis ... | |||
TMPH-01389 | G6PC Protein, Human, Recombinant (His) | Human | Yeast |
Hydrolyzes glucose-6-phosphate to glucose in the endoplasmic reticulum. Forms with the glucose-6-phosphate transporter (SLC37A4/G6PT) the complex responsible for glucose production in the terminal step of glycogenolysis ... | |||
TMPY-05062 | NRG2 Protein, Human, Recombinant (His) | Human | HEK293 |
Neuregulin-2 (NRG2) is a novel member of the neuregulin family of growth and differentiation factors. Through interaction with the ErbB family of receptors, neuregulin-2 induces the growth and differentiation of epitheli... | |||
TMPH-00550 | Epstein-Barr virus (strain B95-8) BCRF1 Protein (His & Myc) | EBV | E. coli |
Plays a role in masking infected cells for immune recognition by cytotoxic T-lymphocytes. Down-regulates the expression of the host TAP1 gene (transporter associated with antigen processing), thereby affecting the transp... | |||
TMPJ-00533 | LYVE1 Protein, Human, Recombinant (His) | Human | Human Cells |
Lymphatic Vessel Endothelial Hyaluronic Acid Receptor 1 is a single-pass type I membrane protein. LYVE-1 is a CD44 homolog found primarily on lymphatic endothelial cells 1. LYVE-1 mainly expressed in endothelial cells li... | |||
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カタログ番号 | 製品名 | ||
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L2550 | Glutamine Metabolism Compound Library | 565 compounds | |
A unique collection of 565 glutamine metabolism related compounds can be used for high throughput screening (HTS) and high content screening (HCS), and also is an effective tool for research in glutamine metabolism and ... |