Powder: -20°C for 3 years | In solvent: -80°C for 1 year
L-803087 is a potent and selective agonist of the growth inhibitor sst4 receptor with a Ki value of 0.7 nM for sst4, which is more than 280-fold more selective than other growth inhibitory receptors.L-803087 induced AMPA-mediated synaptic responses in the hippocampus in vitro, and in vivo increased seizures in alginate-induced seizure-busting mice.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 45,500 | |||
5 mg | 在庫あり | ¥ 123,500 | |||
10 mg | 在庫あり | ¥ 198,000 | |||
25 mg | 在庫あり | ¥ 363,000 | |||
50 mg | 在庫あり | ¥ 636,000 | |||
100 mg | 在庫あり | ¥ 1,017,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 132,500 |
ターゲット&IC50 | SST2 receptor:4720 nM (ki), SST1 receptor:199 nM (ki), SST3 receptor:1280 nM (ki), SST5 receptor:3880 nM (ki), SST4 receptor:0.7 nM (ki) |
分子量 | 485.53 |
分子式 | C25H29F2N5O3 |
CAS No. | 217480-26-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (113.28 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
L-803087 217480-26-7 GPCR/G Protein Somatostatin L 803087 L803087 Inhibitor inhibitor inhibit