Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Monatepil maleate (AJ-2615 maleate) is an orally active Ca2+-channel and α1-adrenoceptor antagonist and non-competitive heparanoyl-coenzyme A:cholesterol acyltransferase (ACAT) inhibitor with antihypertensive activity.Monatepil maleate is used in studies of hyperlipidemia and atherosclerosis. Monatepil maleate is used to study hyperlipidemia and atherosclerosis.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 67,500 |
5 mg | 在庫あり | ¥ 166,000 |
10 mg | 在庫あり | ¥ 226,500 |
25 mg | 在庫あり | ¥ 349,000 |
50 mg | 約6-8 週間 | ¥ 454,500 |
説明 | Monatepil maleate (AJ-2615 maleate) is an orally active Ca2+-channel and α1-adrenoceptor antagonist and non-competitive heparanoyl-coenzyme A:cholesterol acyltransferase (ACAT) inhibitor with antihypertensive activity.Monatepil maleate is used in studies of hyperlipidemia and atherosclerosis. Monatepil maleate is used to study hyperlipidemia and atherosclerosis. |
In vivo | In 8-week-old male Japanese white rabbits (fed with a high cholesterol diet), Monatepil maleate (30 mg/kg; oral administration; once daily for 9 weeks) improved plasma lipid metabolism, reduced atherosclerotic lesions, and lowered blood pressure[1]. |
別名 | AJ2615 maleate, AJ-2615 maleate, AJ 2615 maleate |
分子量 | 591.69 |
分子式 | C32H34FN3O5S |
CAS No. | 103379-03-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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Monatepil maleate 103379-03-9 GPCR/G Protein Membrane transporter/Ion channel Metabolism Neuroscience Adrenergic Receptor Acyltransferase Calcium Channel AJ-2615 AJ2615 maleate AJ-2615 maleate AJ 2615 maleate AJ2615 AJ 2615 Inhibitor inhibitor inhibit