Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC50 = 3 μM).
説明 | BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC50 = 3 μM). |
別名 | BMS 986122 |
分子量 | 448.78 |
分子式 | C16H15BrClNO3S2 |
CAS No. | 313669-88-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (222.83 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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BMS-986122 313669-88-4 Endocrinology/Hormones GPCR/G Protein Neuroscience Opioid Receptor positive BMS 986122 modulator allosteric BMS986122 recruitment β-arrestin adenylyl inhibit cyclase Inhibitor protein inhibitor