keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. Also high affinity CB2 positive allosteric modulator (Ki = 50 nM).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 52,000 |
5 mg | 在庫あり | ¥ 112,000 |
10 mg | 在庫あり | ¥ 163,500 |
25 mg | 在庫あり | ¥ 250,500 |
50 mg | 在庫あり | ¥ 340,000 |
100 mg | 在庫あり | ¥ 454,500 |
500 mg | 在庫あり | ¥ 911,500 |
説明 | RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. Also high affinity CB2 positive allosteric modulator (Ki = 50 nM). |
ターゲット&IC50 | CB2:Ki = 50 nM |
分子量 | 1484.71 |
分子式 | C67H109N19O19 |
CAS No. | TP1939L1 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Insoluble
H2O: 10 mM
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
RVD-Hpα acetate(1193362-76-3 free base) TP1939L1 GPCR/G Protein Cannabinoid Receptor RVD-Hpalpha acetate(1193362-76-3 free base) RVD Hpα acetate(1193362 76 3 free base) RVD-Hpa acetate(1193362-76-3 free base) RVDHpα acetate(1193362763 free base) Inhibitor inhibitor inhibit