Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.
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1 mg | 在庫あり | ¥ 45,500 | |||
2 mg | 在庫あり | ¥ 68,500 | |||
5 mg | 在庫あり | ¥ 108,000 | |||
10 mg | 在庫あり | ¥ 158,000 | |||
25 mg | 在庫あり | ¥ 248,000 | |||
50 mg | 在庫あり | ¥ 333,000 | |||
100 mg | 在庫あり | ¥ 450,000 |
説明 | CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2. |
In vitro | CB2 receptor agonist 2 (compound 4g) (1 μM; 72 hours) shows low or no cytotoxicity to Hep-G2 cells[1]. |
In vivo | CB2 receptor agonist 2 (compound 4g) (1 and 3 mg/kg; 1 hour) is very potent (with maximal effect being reached already at the 1 mg/kg dose) and has antihyperalgesic effects, efficacious also on the first phase of the nocifensive response and strongly reduced by AM630, a CB2-selective antagonist/inverse agonist [1]. |
別名 | ZINC72105556, 4-Quinolone-3-Carboxamide Furan CB2 Agonist |
分子量 | 488.62 |
分子式 | C30H36N2O4 |
CAS No. | 1314230-75-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 3mg/mL (6.1mM)
You can also refer to dose conversion for different animals. 詳細
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CB2 receptor agonist 2 1314230-75-5 GPCR/G Protein Cannabinoid Receptor ZINC72105556 ZINC-72105556 4-Quinolone-3-Carboxamide Furan CB2 Agonist ZINC 72105556 Inhibitor inhibitor inhibit