keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Valorphin TFA(144313-54-2(free base)) is a semisynthetic derivative of dihydrovaltrate with opioid analgesic activity
説明 | Valorphin TFA(144313-54-2(free base)) is a semisynthetic derivative of dihydrovaltrate with opioid analgesic activity |
In vitro | In vitro binding studies using brain homogenates from rat and guinea-pig indicate a preference for the mu-receptor site.?Bath application to cultured cerebellar Purkinje cells inhibited the spontaneous firing, similar to the effect seen with morphine.?Analgesic activity has been demonstrated in the hot plate and the tail flick test in the mouse and the Randall-Selitto test in the rat.?In the rhesus monkey valorphin was self-administered, but naloxone challenge induced only mild withdrawal signs.?Valorphin is a novel chemical entity, structurally not related to known opioids, which interacts preferentially with opiate mu-receptors[1]. |
別名 | Valorphin TFA(144313-54-2(free bas)) |
分子量 | 1006.03 |
分子式 | C46H62F3N9O13 |
CAS No. | T7666 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 10.06 mg/mL (10 mM)
You can also refer to dose conversion for different animals. 詳細
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