Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Enpp-1-IN-14 is a potent inhibitor of Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) with an IC50 value of 32.38 nM for recombinant human ENPP-1.Enpp-1-IN-14 has anti-tumor activity.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 12,000 | |||
5 mg | 在庫あり | ¥ 28,000 | |||
10 mg | 在庫あり | ¥ 45,500 | |||
25 mg | 在庫あり | ¥ 104,500 | |||
50 mg | 在庫あり | ¥ 154,500 | |||
100 mg | 在庫あり | ¥ 219,500 | |||
1 mL * 5 mM (in DMSO) | 在庫あり | ¥ 30,500 |
説明 | Enpp-1-IN-14 is a potent inhibitor of Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) with an IC50 value of 32.38 nM for recombinant human ENPP-1. Enpp-1-IN-14 has anti-tumor activity. |
In vivo | Enpp-1-IN-14 (compound 015) (50 mg/kg; IP; BID, for 31 days) significantly inhibits tumor growth in Female C57BL/6 mice (4-6 weeks; implanted subcutaneously with 2×105 MC38 cells). |
分子量 | 403.88 |
分子式 | C15H22ClN5O4S |
CAS No. | 2687222-59-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 3.33 mg/mL (8.25 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Enpp-1-IN-14 2687222-59-7 Metabolism PDE Inhibitor inhibitor inhibit