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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T35332 | THZ1 2HCl | THZ1 2HCl,THZ1 Dihydrochloride | CDK |
THZ1 2HCl (THZ1 Dihydrochloride) is a selective, covalent, and allosteric inhibitor of CDK7 with an IC50 of 3.2 nM. THZ1 2HCl has antiproliferative effects on a variety of cancer cell lines. | |||
T13153 | THZ1-R | CDK | |
THZ1-R displays diminished activity for CDK7 inhibition(Kd:142 nM). | |||
T72512 | THZ1 Hydrochloride | ||
THZ1 Hydrochloride is a potent, selective covalent inhibitor of CDK7, exhibiting an IC50 value of 3.2 nM. It also targets closely related kinases CDK12 and CDK13, leading to the downregulation of MYC expression. | |||
T3664 | THZ1 | CDK7 inhibitor,THZ1 2HCl | CDK |
THZ1 (CDK7 inhibitor) is a novel selective and potent covalent CDK7 inhibitor. |