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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T15737 | Lesogaberan | AZD-3355 | GABA Receptor |
Lesogaberan is an effective and selective GABAB receptor agonist (EC50: 8.6 nM for human recombinant GABAB receptors). For rat brain GABAB and GABAA receptors, the binding affinity (Kis) is 5.1 nM and 1.4 μM, respectivel... |