GABA Receptor

The GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels (also known as ionotropic receptors); whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors.

Cat. No.	製品名	CAS No.	Purity
T21793	CGP 35348	123690-79-9	98%
T21793	CGP 35348 is a selective antagonist of GABAB receptor (EC50 = 34 μM). CGP 35348 can be used in studies of neuromuscular coordination and spatial learning after n...
T28479	PZ-II-029	164025-44-9	98%
T28479	PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.
T4522	SSD114 hydrochloride	T4522	98%
T4522	SSD114 is a novel GABAB receptor positive allosteric modulator.
T8193	α-Thujone	546-80-5	98%
T8193	Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.
T16539	Piperazine citrate	144-29-6	98%
T16539	Piperazine Citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring. It used as an Anthelmi...
T8268	6,2'-Dihydroxyflavone	92439-20-8	98%
T8268	6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.
T32098L	Homocarnosine acetate		98%
T32098L	Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine. Homocarnosine acetate has antioxidant and anti-infla...
T2407	Tiagabine	115103-54-3	98%
T2407	Tiagabine is an Anti-epileptic Agent. The physiologic effect of tiagabine is by means of Decreased Central Nervous System Disorganized Electrical Activity.
T37190	L-Allylglycine	16338-48-0	98%
T37190	L-Allylglycine is an amino acid derivative that reduces glutamate decarboxylase (GAD) activity by 60% when administered at a dose of 39.8 μmol/g per hour ex vivo...
T1240	Flumazenil	78755-81-4	98%
T1240	Flumazenil antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous system (CNS),...
T5880	Aminooxyacetic acid hemihydrochloride	2921-14-4	98%
T5880	Aminooxyacetic acid hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T.
T3782	Jujuboside A	55466-04-1	98%
T3782	Jujuboside A is a glycoside extracted from Semen Ziziphi Spinosae, having neurophysiological inhibitory effects, used as a potential therapeutic agent for the tr...
T3173	DAA-1106	220551-92-8	98%
T3173	DAA1106 is a potent and selective ligand for peripheral benzodiazepine receptor (PBR), acting as a potent and selective agonist at the peripheral benzodiazepine ...
T0024	Primidone	125-33-7	98%
T0024	Primidone is an anticonvulsant of the pyrimidinedione class.
T3644	U93631	152273-12-6	98%
T3644	GABAA receptor antagonist that binds the picrotoxin site and stabilizes the inactive form of the channel via allosteric interaction. Accelerates the decay of GAB...
T22616	Bretazenil	84379-13-5	98%
T22616	GABAA benzodiazepine site partial agonist
T4993	Afloqualone	56287-74-2	98%
T4993	Afloqualone is a agonist of GABA Receptor . Target: GABA Receptor in vitro: Afloqualone is a quinazolinone family GABAergic drug. It has sedative and muscle-rela...
T0715	Chlormezanone	80-77-3	98%
T0715	Chlormezanone is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.
T9424	Temgicoluril	10095-06-4	98%
T9424	Temgicoluril acts on GABA Receptor.
T0675	Topiramate	97240-79-4	98%
T0675	Topiramate is a unique antiseizure medication that is used in the treatment of partial and generalized seizures. Topiramate has been rarely associated with hepat...