| T21793 |
CGP 35348
|
123690-79-9
|
98%
|
|
|
CGP 35348 is a selective antagonist of GABAB receptor (EC50 = 34 μM). CGP 35348 can be used in studies of neuromuscular coordination and spatial learning after n...
|
| T28479 |
PZ-II-029
|
164025-44-9
|
98%
|
|
|
PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.
|
| T8268 |
6,2'-Dihydroxyflavone
|
92439-20-8
|
98%
|
|
|
6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.
|
| T32098L |
Homocarnosine acetate
|
|
98%
|
|
|
Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine. Homocarnosine acetate has antioxidant and anti-infla...
|
| T37190 |
L-Allylglycine
|
16338-48-0
|
98%
|
|
|
L-Allylglycine is an amino acid derivative that reduces glutamate decarboxylase (GAD) activity by 60% when administered at a dose of 39.8 μmol/g per hour ex vivo...
|
| T4S1616 |
Sanggenon D
|
81422-93-7
|
98%
|
|
|
Sanggenone D represents a new scaffold of positive GABAA receptor modulators, it also inhibits COX-2 activity (IC 50 = 73-100 μM). Sanggenone D has anti-inflamma...
|
| T1240 |
Flumazenil
|
78755-81-4
|
98%
|
|
|
Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous ...
|
| T4993 |
Afloqualone
|
56287-74-2
|
98%
|
|
|
Afloqualone (HQ-495) is a agonist of GABA Receptor . Target: GABA Receptor in vitro: Afloqualone is a quinazolinone family GABAergic drug. It has sedative and mu...
|
| TN1308 |
6-Hydroxyflavanone
|
4250-77-5
|
98%
|
|
|
6-Hydroxyflavanone, extracted from the leaves of Acorus calamus, exhibits anti-inflammatory and anti-neuropathic pain activity by targeting cyclooxygenase-2 (COX...
|
| T24381 |
L-822179
|
215874-86-5
|
98%
|
|
|
L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.
|
| T16489 |
Darigabat
|
1614245-70-3
|
98%
|
|
|
Darigabat (PF-06372865) is an orally active and selective GABAA receptor modulator that crosses the blood-brain barrier and exhibits anxiolytic activity, with Ki...
|
| T2998 |
Dihydromyricetin
|
27200-12-0
|
|
|
|
Dihydromyricetin (Ampelopsin) is a natural antioxidant flavonoid from Ampelopsis grossedentata. Dihydromyricetin is a potent inhibitor of dihydropyrimidinase wit...
|
| T16539 |
Piperazine citrate
|
144-29-6
|
|
|
|
Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring. It used as an Anthelmi...
|
| T5880 |
Aminooxyacetic acid hemihydrochloride
|
2921-14-4
|
|
|
|
Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degrada...
|
| T12492 |
Pivagabine
|
69542-93-4
|
|
|
|
Pivagabine (CXB-722), a hydrophobic 4-aminobutyric acid derivative, exhibits neuromodulatory activity and successfully penetrates the blood-brain barrier in rats...
|
| T1673 |
Acamprosate calcium
|
77337-73-6
|
|
|
|
Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.
|
| T20657 |
Muscimol HBr
|
18174-72-6
|
100%
|
|
|
Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.
|
| T27845 |
Losigamone
|
112856-44-7
|
100%
|
|
|
Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.
|
| T26834 |
BL-1020 Mesylate
|
916898-61-8
|
100%
|
|
|
BL-1020 Mesylate (CYP-1020 Mesylate) is an orally available GABA A receptor agonist and D2 antagonist that decreases dopamine activity and enhances GABAA activit...
|
| T8568 |
Suritozole
|
110623-33-1
|
100%
|
|
|
Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptor
|
