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Search Results for " 5‐HT1C "

ターゲット

Potassium Channel Dopamine Receptor 5-HT Receptor

阻害剤

天然化合物

リコンビナントタンパク質

カタログ番号	製品名	別名	ターゲット
T4369	SCH-23390 hydrochloride	R-(+)-SCH23390 hydrochloride	Potassium Channel , Dopamine Receptor , 5-HT Receptor
	SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).		Potassium Channel , Dopamine Receptor , 5-HT Receptor
T12865	SCH-23390 maleate	R-(+)-SCH-23390 maleate	Potassium Channel , Dopamine Receptor , 5-HT Receptor
			Potassium Channel , Dopamine Receptor , 5-HT Receptor
T22689	CP94253 hydrochloride	CP 94253 hydrochloride	Others , 5-HT Receptor
	CP94253 hydrochloride (CP 94253 hydrochloride) is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, ...		Others , 5-HT Receptor
T5389	Volinanserin	M 100907,MDL100907	5-HT Receptor
	Volinanserin (MDL100907) (MDL 100907) is a potent and selective antagonist of the serotonin receptor 5-HT2 (Ki: 0.36 nM) and shows 300-fold selectivity for 5-HT2 receptor over 5-HT1c, alpha-1 adrenergic and sigma recepto...		5-HT Receptor
T0225	Pizotifen Malate	Pizotyline (malate),BC-105 (malate),BC-105	5-HT Receptor
	Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based on benzocycloheptane.		5-HT Receptor
T22987	MK 212 hydrochloride		5-HT Receptor
	MK 212 hydrochloride is a 5-HT2C receptor agonist		5-HT Receptor
T1442	Pizotifen	Pizotyline,BC-105	5-HT Receptor
	Pizotifen (Pizotyline) is a strong serotonin and tryptamine antagonist, with weak anticholinergic, anti-histaminic and anti-kinin effects. It also possesses sedative and appetite-stimulating properties. Pizotifen hydroch...		5-HT Receptor
T28637	S 14506 HCl	S14506 HCl,S-14506,S14506HCl
	S 14506 HCl is a highly potent selective 5-HT1A receptor full agonist, pKi values are 9.0, 6.6, 7.5, 6.6 and < 6.0 for 5-HT1A, 5-HT1B, 5-HT1C, 5-HT2 and 5-HT3 receptors respectively.
T27574	ZM 169369	ICI169369,ICI-169369
	ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.
T3046	BMY 7378 dihydrochloride	BMY7378 HCl	Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
	BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.		Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor

Compounds

SCH-23390 hydrochloride

T4369

Synonym: R-(+)-SCH23390 hydrochloride

Target: Potassium Channel, Dopamine Receptor, 5-HT Receptor

SCH-23390 maleate

T12865

Synonym: R-(+)-SCH-23390 maleate

Target: Potassium Channel, Dopamine Receptor, 5-HT Receptor

CP94253 hydrochloride

T22689

Synonym: CP 94253 hydrochloride

Target: Others, 5-HT Receptor

Volinanserin

T5389

Synonym: M 100907,MDL100907

Target: 5-HT Receptor

Pizotifen Malate

T0225

Synonym: Pizotyline (malate),BC-105 (malate),BC-105

Target: 5-HT Receptor

MK 212 hydrochloride

T22987

Synonym:

Target: 5-HT Receptor

Pizotifen

T1442

Synonym: Pizotyline,BC-105

Target: 5-HT Receptor

S 14506 HCl

T28637

Synonym: S14506 HCl,S-14506,S14506HCl

Target:

ZM 169369

T27574

Synonym: ICI169369,ICI-169369

Target:

BMY 7378 dihydrochloride

T3046

Synonym: BMY7378 HCl

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor

カタログ番号	製品名	別名	ターゲット
T1045	Trimipramine maleate	Surmontil maleate	Dopamine Receptor , 5-HT Receptor , Antibacterial , Adrenergic Receptor , Norepinephrine , Histamine Receptor
	Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Mal...
T21855	AMI-193	Espiramida,Spiramide	Dopamine Receptor , 5-HT Receptor
	AMI-193 (Spiramide) is an effective and selective antagonist of 5-HT2 and D2 receptor with Kis of 2, 3, 50, 2530, and 4300 nM for 5-HT2, D2 Receptor, 5-HT1A, D1 Receptor, and 5-HT1C Receptor. AMI-193 shows antipsychotic ...		Dopamine Receptor , 5-HT Receptor

天然物製品

Trimipramine maleate

T1045

Synonym: Surmontil maleate

Target: Dopamine Receptor, 5-HT Receptor, Antibacterial, Adrenergic Receptor, Norepinephrine, Histamine Receptor

AMI-193

T21855

Synonym: Espiramida,Spiramide

Target: Dopamine Receptor, 5-HT Receptor

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-05308	CD45 Protein, Human, Recombinant (aa 1-529, His)	Human	HEK293 Cells
	CD45 Protein, Human, Recombinant (aa 1-529, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 57.4 kDa and the accession number is P08575-5.
TMPJ-00854	ETS1 Protein, Human, Recombinant (His)	Human	E. coli
	ETS1 Protein (ETS1) is a nuclear protein that belongs to the ETS family. Members of this family recognize the core consensus DNA sequence GGAA/T in target genes. Proteins function either as transcriptional activators or ...
TMPY-05498	SR-BI/SCARB1 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	SR-BI/SCARB1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 73.4 kDa and the accession number is Q8WTV0-5.
TMPY-05387	SLAMF7 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	SLAMF7 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 49.1 kDa and the accession number is Q9NQ25-5.
TMPY-05547	SLAMF7 Protein, Human, Recombinant (hFc), Biotinylated	Human	HEK293 Cells
	SLAMF7 Protein, Human, Recombinant (hFc), Biotinylated is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 49.1 kDa and the accession number is Q9NQ25-5.
TMPY-04318	GRIK2 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	GRIK2 (Glutamate Ionotropic Receptor Kainate Type Subunit 2, also known as GluR6) is a Protein Coding gene. The GRIK2 (one of the kainate receptors) gene resides in a genetic linkage region (6q21) associated with bipolar...
TMPK-01363	SIRP alpha V5 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	Signal regulatory protein α (SIRPα) is a regulatory membrane glycoprotein from SIRP family expressed mainly by myeloid cells and also by stem cells or neurons.SIRPα acts as inhibitory receptor and interacts with a broadl...
TMPK-01357	SIRP alpha V5 Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	Signal regulatory protein α (SIRPα) is a regulatory membrane glycoprotein from SIRP family expressed mainly by myeloid cells and also by stem cells or neurons.SIRPα acts as inhibitory receptor and interacts with a broadl...